Regulation of opioid receptor function by chronic agonist exposure: Constitutive activity and desensitization

被引：58

作者：

Chavkin, C ^{[1
]}

McLaughlin, JP ^{[1
]}

Celver, JP ^{[1
]}

机构：

[1] Univ Washington, Hlth Sci Ctr, Dept Pharmacol, Seattle, WA 98195 USA

来源：

MOLECULAR PHARMACOLOGY | 2001年 / 60卷 / 01期

关键词：

D O I：

10.1124/mol.60.1.20

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

[No abstract available]

引用

页码：20 / 25

页数：6

共 56 条

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[9] Threonine 180 is required for G-protein-coupled receptor kinase 3- and β-arrestin 2-mediated desensitization of the μ-opioid receptor in Xenopus oocytes
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