Solvent-free Pd-catalysed N-arylation of amines, amides and diaza-18-crown-6

被引：20

作者：

Artamkina, GA ^{[1
]}

Ermolina, MV ^{[1
]}

Beletskaya, IP ^{[1
]}

机构：

[1] Moscow MV Lomonosov State Univ, Dept Chem, Moscow 119992, Russia

来源：

MENDELEEV COMMUNICATIONS | 2003年 / 04期

基金：

俄罗斯基础研究基金会;

关键词：

D O I：

10.1070/MC2003v013n04ABEH001753

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

The N-arylation of amines, amides and diaza-18-crown-6 with-weakly activated aryl bromides catalysed by (PdL)-L-0 and the arylation of pyrrolidone-2 with 2-bromothiophene catalysed by CuI/1,2-di(methylamino)cyclohexane can be performed in the presence of graphite at 60-100degreesC without solvent to give arylation products in good yields (60-78%).

引用

页码：158 / 160

页数：3

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