A highly useful method for the acylation of amines with acid chlorides utilizing sodium 2-ethylhexanoate as the base is described. This procedure is superior to the Schonen-Baumann conditions whenever the product is water soluble. (C) 1998 Elsevier Science Ltd. All rights reserved.
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页码:6991 / 6992
页数:2
相关论文
共 3 条
[1]
CABRE J, 1997, Patent No. 9715579
[2]
NYCE PL, 1991, SYNTHESIS-STUTTGART, P571
[3]
Pessa A., 1997, U.S. Patent, Patent No. [5,625,058, 5625058]