Microwave induced synthesis of 2-substituted phenyl-3-(3-alkyl/aryl-5,6-dihydro-S-triazolo)[2,4-B][1,3,4]thiadiazo 6-yl indoles and 2-phenyl-3 [2,substituted benzothiazole] derivatives and their fungicidal activity

被引:8
作者
Dandia, A [1 ]
Rani, B
Saha, M
Gupta, IJ
机构
[1] Univ Rajasthan, Dept Chem, Jaipur 302004, Rajasthan, India
[2] Rajasthan Agr Univ, Agr Res Stn, Seed Technol Res Ctr, Jaipur 302018, Rajasthan, India
来源
PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS | 1997年 / 130卷
关键词
sulfur-containing indole derivatives; 4-amino-5-mercaptotriazole; 2-aminothiophenol; benzothiazole; triazolothiadiazoles; microwave irradiation; antifungal activity; ANTIBACTERIAL ACTIVITY; ORGANIC-SYNTHESIS; CHEMISTRY; FLUORINE; OVENS; SPIROHETEROCYCLES; 1,2,4-TRIAZOLES; AGENTS;
D O I
10.1080/10426509708033712
中图分类号
O61 [无机化学];
学科分类号
070301 ; 081704 ;
摘要
The title compounds were synthesised by condensation of 3-alykl/aryl-4-amino-5-mercaptotriazole (II) and 5-substituted 2-aminothiophenols (IV) with appropriate 2-phenyl-1H-indole-3-carboxaldehyde (I) under microwave irradiation in the presence of piperidine/p-toluenesulphonic acid using ethanol/DMF as energy transfer media. The considerable increase in reaction rare with improved yield has been observed, using microwave as compared to classical method.
引用
收藏
页码:217 / 227
页数:11
相关论文
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