A straightforward route to 4H-1,4-benzoxazine-2-carbaldehydes by Swern oxidation

被引：13

作者：

Bourlot, AS

Guillaumet, G

Merour, JY

机构：

[1] Lab. de Chim. Bioorgan./Analytique, URA CNRS No. 499, Université d'Orléans, 45067 Orléans Cedex 2

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 1996年 / 33卷 / 01期

关键词：

D O I：

10.1002/jhet.5570330133

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Swern oxidation of saturated (1,4-benzoxazine-2-yl)-methanols 2 furnished 4H-1,4-benzoxazine-2-carbaldehydes 3, which possess an alpha,beta ethylenic bond. The reactivity of these compounds was examined.

引用

页码：191 / 196

页数：6

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