Discovery and optimization of a novel series of thrombin receptor (PAR-1) antagonists: Potent, selective peptide mimetics based on indole and indazole templates

被引：75

作者：

Zhang, HC ^{[1
]}

Derian, CK

Andrade-Gordon, P

Hoekstra, WJ

McComsey, DF

White, KB

Poulter, BL

Addo, MF

Cheung, WM

Damiano, BP

Oksenberg, D

Reynolds, EE

Pandey, A

Scarborough, RM

Maryanoff, BE

机构：

[1] RW Johnson Pharmaceut Res Inst, Spring House, PA 19477 USA

[2] COR Therapeut Inc, S San Francisco, CA 94080 USA

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 2001年 / 44卷 / 07期

关键词：

D O I：

10.1021/jm000506s

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1021 / 1024

页数：4

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