Design, synthesis and biological activity of novel enediynyl monocyclic beta-lactams

被引：19

作者：

Basak, A

Khamrai, UK

机构：

[1] Department of Chemistry, Indian Institute of Technology

来源：

TETRAHEDRON LETTERS | 1996年 / 37卷 / 14期

关键词：

D O I：

10.1016/0040-4039(96)00297-3

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Monocyclic beta-lactams 1-3 substituted at C-4 with enediyne moiety have been synthesized via Pd(0) mediated coupling reaction. Their antibacterial activity against ampicillin-resistant E. coli have been tested. Copyright (C) 1996 Published by Elsevier Science Ltd.

引用

页码：2475 / 2478

页数：4

共 18 条

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