Direct arylations on water: synthesis of 2,5-disubstituted oxazoles balsoxin and texaline

被引:148
作者
Ohnmacht, Stephan A. [1 ]
Mamone, Patrizia [1 ]
Culshaw, Andrew J. [2 ]
Greaney, Michael F. [1 ]
机构
[1] Univ Edinburgh, Sch Chem, Edinburgh EH9 3JJ, Midlothian, Scotland
[2] Novartis Horsham Res Ctr, Global Discovery Chem, Horsham RH12 5AB, W Sussex, England
关键词
D O I
10.1039/b719466h
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
An efficient two-step palladium catalysed synthesis of 2,5-disubstituted oxazoles is reported.
引用
收藏
页码:1241 / 1243
页数:3
相关论文
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