A convenient method for the synthesis of 2-trichloromethyl-4-p-substituted-phenyl-3H-1,5-benzodiazepines.

被引：56

作者：

Bonacorso, HG

Bittencourt, ST

Wastowski, AD

Wentz, AP

Zanatta, N

Martins, MAP

机构：

[1] Departamento de Química, Univ. Federal de Santa Maria(UFSM), 97119-900 Santa Maria, RS

来源：

TETRAHEDRON LETTERS | 1996年 / 37卷 / 51期

关键词：

D O I：

10.1016/S0040-4039(96)02145-4

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A convenient method to obtain a new series of 2-trichloromethyl-4-aryl-3H-1,5-benzodiazepines from the reaction of beta-methoxyvinyl trichloromethyl ketones derived from acetals and o-phenylenediamine is reported. Copyright (C) 1996 Elsevier Science Ltd

引用

页码：9155 / 9156

页数：2

共 8 条

[1]

CHIMIRRI A, 1993, HETEROCYCLES, V36, P3

[2]

KATRITZKY AR, 1984, COMPREHENSIVE HETERO, V7, P594

[3]

Lloyd D., 1974, ADV HETEROCYCLIC CHE, V17, P27

[4] Heterocyclic variants of 1,5-benzodiazepine system .7. Synthesis of substituted 2a-phenyl-4-methylsulfonyl-2-methoxy-1,2,2a,3-tetrahydroazeto[1,2-a][1,5]benzodiazepin-1-ones [J].