Flubendiamide, a novel insecticide highly active against lepidopterous insect pests

被引:290
作者
Tohnishi, M
Nakao, H
Furuya, T
Seo, A
Kodama, H
Tsubata, K
Fujioka, S
Kodama, H
Hirooka, T
Nishimatsu, T
机构
[1] Nihon Nohyaku Co Ltd, Res Ctr, Osaka 5860094, Japan
[2] Nihon Nohyaku Co Ltd, Div Res & Dev, R&D Strategy Dept, Chuo Ku, Tokyo 1038236, Japan
[3] Nihon Nohyaku Co Ltd, Sales Div, Mkt & Sales Dept, Chuo Ku, Tokyo 1038236, Japan
关键词
benzenedicarboxamide; flubendiamide; heptafluoroisopropylanilide; insecticide; lepidoptericide;
D O I
10.1584/jpestics.30.354
中图分类号
Q96 [昆虫学];
学科分类号
摘要
Flubendiamide, N-2-[1, 1-dimethyl-2-(methylsulfonyl)ethyl]-3-iodo-N-1-[2-methyl-4-[1,2,2,2-tetrafluoro-1-(trifluoromethyl)ethyl]phenyl]-1,2-benzenedicarboxamide.. is a novel class of insecticide having a unique chemical structure. The uniqueness of the structure results from three parts with novel substituents; a heptafluoroisopropyl group in the anilide moiety, a sulfonylalkyl group in the aliphatic amide moiety, and an iodine atom at the 3-position of the phthalic acid moiety. The compound shows extremely strong insecticidal activity especially against lepidopterous pests including resistant strains. Flubendiamide would have a novel mode of action, because the insecticidal symptoms accompanied by a discriminative contraction of the larval body are distinguished from those of commercial insecticides. It is also very safe for non-target organisms. Flubendiamide is expected to be a suitable agent for controlling lepidopterous insects as part of the insect resistance management and the integrated pest management programs. (c) Pesticide Science Society of Japan.
引用
收藏
页码:354 / 360
页数:7
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