A new approach to the synthesis of non-racemic isoindolin-1-one derivatives

被引：34

作者：

Allin, SM

Northfield, CJ

Page, MI ^{[1
]}

Slawin, AMZ

机构：

[1] Loughborough Univ Technol, Dept Chem, Loughborough LE11 3TU, Leics, England

[2] Univ Huddersfield, Dept Chem & Biol Sci, Huddersfield HD1 3DH, W Yorkshire, England

来源：

TETRAHEDRON LETTERS | 1999年 / 40卷 / 01期

关键词：

amino alcohols; aminals; stereocontrol; transition states; nitrogen heterocycles;

D O I：

10.1016/S0040-4039(98)80041-5

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A new approach for the synthesis of non-racemic 3-substituted isoindolin-1-one targets has been developed through application of a tricyclic gamma-lactam substrate as an N-acyliminium ion precursor. (C) 1998 Elsevier Science Ltd. All rights reserved.

引用

页码：141 / 142

页数：2

共 9 条

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