On the cyclization of acyliminium salts derived from pyroglutamic acid.

被引：22

作者：

Rigo, B ^{[1
]}

ElGhammarti, S ^{[1
]}

Couturier, D ^{[1
]}

机构：

[1] UNIV SCI & TECHNOL LILLE,F-59655 VILLENEUVE DASCQ,FRANCE

来源：

TETRAHEDRON LETTERS | 1996年 / 37卷 / 04期

关键词：

D O I：

10.1016/0040-4039(95)02215-5

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The Friedel Crafts reaction of pyroglutamic acid derivative 9 gives an acyliminium salt which cyclize to the condensed N-acylheterocycle 6 thus providing an easy access to the amine 1.

引用

页码：485 / 486

页数：2

共 12 条

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