The human keratinocyte cell line HaCaT: An in vitro cell culture model for keratinocyte testosterone metabolism

被引:19
作者
Altenburger, R [1 ]
Kissel, T [1 ]
机构
[1] Univ Marburg, Dept Pharmaceut & Biopharm, Marburg, Germany
关键词
cell culture; keratinocytes; androgen metabolism; testosterone; transdermal delivery; 5; alpha-reductase;
D O I
10.1023/A:1011945212831
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
[No abstract available]
引用
收藏
页码:766 / 771
页数:6
相关论文
共 15 条
[1]  
ALTENBURGER R, IN PRESS PHARM RES
[2]   LACTATE-DEHYDROGENASE RELEASE AS AN INDICATOR OF DITHRANOL-INDUCED MEMBRANE INJURY IN CULTURED HUMAN KERATINOCYTES - A TIME PROFILE STUDY [J].
BONNEKOH, B ;
FARKAS, B ;
GEISEL, J ;
MAHRLE, G .
ARCHIVES OF DERMATOLOGICAL RESEARCH, 1990, 282 (05) :325-329
[3]   NORMAL KERATINIZATION IN A SPONTANEOUSLY IMMORTALIZED ANEUPLOID HUMAN KERATINOCYTE CELL-LINE [J].
BOUKAMP, P ;
PETRUSSEVSKA, RT ;
BREITKREUTZ, D ;
HORNUNG, J ;
MARKHAM, A ;
FUSENIG, NE .
JOURNAL OF CELL BIOLOGY, 1988, 106 (03) :761-771
[4]   The 5 alpha-reductase system and its inhibitors - Recent development and its perspective in treating androgen-dependent skin disorders [J].
Chen, W ;
Zouboulis, CC ;
Orfanos, CE .
DERMATOLOGY, 1996, 193 (03) :177-184
[5]   MK386: A potent, selective inhibitor of the human type 1 5 alpha-reductase [J].
Ellsworth, K ;
Azzolina, B ;
Baginsky, W ;
Bull, H ;
Chang, B ;
Cimis, G ;
Mitra, S ;
Toney, J ;
Bakshi, RK ;
Rasmusson, GR ;
Tolman, RL ;
Harris, GS .
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 1996, 58 (04) :377-384
[6]   ABSORPTION AND METABOLISM OF TOPICALLY APPLIED TESTOSTERONE IN AN ORGANOTYPIC SKIN CULTURE [J].
ERNESTI, AM ;
SWIDEREK, M ;
GAY, R .
SKIN PHARMACOLOGY, 1992, 5 (03) :146-153
[7]  
GORMAR FE, 1993, CELL TISSUE CULTURE, P126
[8]  
HOTCHKISS SAM, 1992, PROGR DRUG METABOLIS, P217
[9]  
LOWRY OH, 1951, J BIOL CHEM, V193, P265
[10]   AZASTEROIDS AS INHIBITORS OF TESTOSTERONE 5-ALPHA-REDUCTASE IN MAMMALIAN SKIN [J].
MELLIN, TN ;
BUSCH, RD ;
RASMUSSON, GH .
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 1993, 44 (02) :121-131