Facile palladium-catalysed synthesis of 1-aryl-1H-indazoles from 2-bromobenzaldehydes and arylhydrazines

被引：83

作者：

Cho, CS ^{[1
]}

Lim, DK

Heo, NH

Kim, TJ

Shim, SC

机构：

[1] Kyungpook Natl Univ, Res Inst Ind Technol, Taegu 702701, South Korea

[2] Kyungpook Natl Univ, Coll Engn, Dept Ind Chem, Taegu 702701, South Korea

来源：

CHEMICAL COMMUNICATIONS | 2004年 / 01期

关键词：

D O I：

10.1039/b312154m

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

2-Bromobenzaldehydes react with arylhydrazines in toluene at 100 degreesC in the presence of a catalytic amount of a palladium catalyst and phosphorus chelating ligands such as 1,1'-bis(diphenylphosphino)ferrocene and 1,3-bis(diphenylphosphino)propane along with NaO-t-Bu to afford 1-aryl-1H-indazoles in good yields.

引用

页码：104 / 105

页数：2

共 20 条

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