Synthesis of substituted 3-trifluoromethylbenzo[b]thiophenes

被引：21

作者：

Owton, WM ^{[1
]}

机构：

[1] Eli Lilly & Co, Lilly Res Ctr Ltd, Windlesham GU20 6PH, Surrey, England

来源：

TETRAHEDRON LETTERS | 2003年 / 44卷 / 38期

关键词：

lithiation; trifluoromethylbenzothiophenes;

D O I：

10.1016/S0040-4039(03)01811-2

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A straightforward method for the synthesis of 5/6-substituted 3-trifluoromethylbenzo[b]thiophenes and their precursor o-fluorinated trifluoro acetophenones is reported. (C) 2003 Elsevier Ltd. All rights reserved.

引用

页码：7147 / 7149

页数：3

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