One-pot synthesis of substituted quinazolin-4(3H)-ones under microwave irradiation

被引：27

作者：

Rad-Moghadam, K ^{[1
]}

Khajavi, MS ^{[1
]}

机构：

[1] Shahid Beheshti Univ, Dept Chem, Tehran 19839, Iran

来源：

JOURNAL OF CHEMICAL RESEARCH-S | 1998年 / 11期

关键词：

D O I：

10.1039/a802853b

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

Synthesis of the title compounds by cyclocondensation of anthranilic acid, formic acid (or orthoesters) and an amine in one pot under microwave irradiation takes place in a few minutes.

引用

页码：702 / 703

页数：3

共 15 条

[1] AN ANTIMALARIAL ALKALOID FROM HYDRANGEA .18. DERIVATIVES OF 4-PYRIMIDONE [J].

BAKER, BR ;

SCHAUB, RE ;

JOSEPH, JP ;

MCEVOY, FJ ;

WILLIAMS, JH .

JOURNAL OF ORGANIC CHEMISTRY, 1953, 18 (02) :133-137

[2] NMR-STUDIES OF 4(3H)-QUINAZOLINONES AND 4(3H)-QUINAZOLINETHIONES [J].

CHAKRABARTY, M ;

BATABYAL, A ;

MORALESRIOS, MS ;

JOSEPHNATHAN, P .

MONATSHEFTE FUR CHEMIE, 1995, 126 (6-7) :789-794

[3] ACYLANTHRANILS .4. EFFECT OF STERIC HINDRANCE ON SELECTIVITY IN REACTION OF AMINES WITH ACETYLANTHRANIL [J].

ERREDE, LA ;

MCBRADY, JJ ;

OIEN, HT .

JOURNAL OF ORGANIC CHEMISTRY, 1977, 42 (04) :656-658

[4]

GRAVIER D, 1992, PHARMAZIE, V47, P91

[5]

HURMER R, 1967, Patent No. 1093977

[6]

JANIAK S, 1969, Patent No. 1908097

[7] Reaction of anthranilic acid with orthoesters: a new facile one-pot synthesis of 2-substituted 4H-3,1-benzoxazin-4-ones [J].

Khajavi, MS ;

Montazari, N ;

Hosseini, SSS .

JOURNAL OF CHEMICAL RESEARCH-S, 1997, (08) :286-287

[8] SYNTHESIS OF 3-AMINO-4(3H)-QUINAZOLINONES FROM N-(2-CARBOMETHOXYPHENYL) IMIDATE ESTERS [J].

LEIBY, RW .

JOURNAL OF ORGANIC CHEMISTRY, 1985, 50 (16) :2926-2929

[9]

MEYER KH, 1943, J ORG CHEM, V8, P239

[10] ROLE OF ALKYL SUBSTITUTION IN 2,3-DISUBSTITUTED AND 3-SUBSTITUTED 4-QUINAZOLONES ON INHIBITION OF PYRUVIC ACID OXIDATION [J].

PARMAR, SS ;

KISHOR, K ;

SETH, PK ;

ARORA, RC .

JOURNAL OF MEDICINAL CHEMISTRY, 1969, 12 (01) :138-&

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