Relative bioavailability of Neoral versus Sandimmune in the presence of a P450IIIA and P-glycoprotein inhibitor

被引:9
作者
Choc, MG [1 ]
Mueller, EA
Robinson, WT
Kumle, A
Smith, HT
Charnick, SB
机构
[1] Nova Pharmaceut Corp, E Hanover, NJ 07936 USA
[2] Novartis Pharma AG, Basel, Switzerland
关键词
D O I
10.1016/S0041-1345(98)00383-2
中图分类号
R392 [医学免疫学]; Q939.91 [免疫学];
学科分类号
100102 ;
摘要
引用
收藏
页码:1664 / 1665
页数:2
相关论文
共 6 条
[1]   Intestinal drug metabolism and antitransport processes: A potential paradigm shift in oral drug delivery [J].
Benet, LZ ;
Wu, CY ;
Hebert, MF ;
Wacher, VJ .
JOURNAL OF CONTROLLED RELEASE, 1996, 39 (2-3) :139-143
[2]   CYCLOSPORINE DISPOSITION AND METABOLITE PROFILES IN RENAL-TRANSPLANT PATIENTS RECEIVING A MICROEMULSION FORMULATION [J].
KOVARIK, JM ;
VERNILLET, L ;
MUELLER, EA ;
FREIBURGHAUS, R ;
NIEDERBERGER, W ;
KUTZ, K .
THERAPEUTIC DRUG MONITORING, 1994, 16 (05) :519-525
[3]  
Meinzer Armin, 1996, P259
[4]  
REYMOND JP, 1988, PHARMACEUT RES, V5, P677, DOI 10.1023/A:1015939307478
[5]   ENHANCED INTESTINAL-ABSORPTION OF CYCLOSPORINE IN RATS THROUGH THE REDUCTION OF EMULSION DROPLET SIZE [J].
TARR, BD ;
YALKOWSKY, SH .
PHARMACEUTICAL RESEARCH, 1989, 6 (01) :40-43
[6]   DIFFERENTIATION OF ABSORPTION AND FIRST-PASS GUT AND HEPATIC-METABOLISM IN HUMANS - STUDIES WITH CYCLOSPORINE [J].
WU, CY ;
BENET, LZ ;
HEBERT, MF ;
GUPTA, SK ;
ROWLAND, M ;
GOMEZ, DY ;
WACHER, VJ .
CLINICAL PHARMACOLOGY & THERAPEUTICS, 1995, 58 (05) :492-497