Efficient synthesis of the 5-HT2c receptor agonist, Org 37684

被引:9
作者
Adams, DR [1 ]
Duncton, MAJ [1 ]
机构
[1] Cerebrus Ltd, Wokingham RG41 5UA, England
关键词
D O I
10.1081/SCC-100104420
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
An efficient synthesis of the 5-HT2C receptor agonist Org 37684 is presented. The synthesis utilises the regioselective demethylation of an arylether as the key step.
引用
收藏
页码:2029 / 2036
页数:8
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