Efficient solid-phase synthesis of diverse 2-aminoquinazolin-4-ones from resin-bound anilines

被引:19
作者
Makino, S [1 ]
Okuzumi, T [1 ]
Tsuji, T [1 ]
Nakanishi, E [1 ]
机构
[1] Ajinomoto Co Inc, Pharmaceut Res Labs, Kawasaki Ku, Kawasaki, Kanagawa 2108681, Japan
来源
JOURNAL OF COMBINATORIAL CHEMISTRY | 2003年 / 5卷 / 06期
关键词
D O I
10.1021/cc030033l
中图分类号
O69 [应用化学];
学科分类号
081704 [应用化学];
摘要
[No abstract available]
引用
收藏
页码:756 / 759
页数:4
相关论文
共 30 条
[1]
Solid-phase organic reactions III: A review of the literature Nov 96 Dec 97 [J].
Booth, S ;
Hermkens, PHH ;
Ottenheijm, HCJ ;
Rees, DC .
TETRAHEDRON, 1998, 54 (51) :15385-15443
[2]
The recent impact of solid-phase synthesis on medicinally relevant benzoannelated nitrogen heterocycles [J].
Bräse, S ;
Gil, C ;
Knepper, K .
BIOORGANIC & MEDICINAL CHEMISTRY, 2002, 10 (08) :2415-2437
[3]
A POTENT, ORALLY-ACTIVE, BALANCED AFFINITY ANGIOTENSIN-II AT(1) ANTAGONIST AND AT(2) BINDING INHIBITOR [J].
DELASZLO, SE ;
QUAGLIATO, CS ;
GREENLEE, WJ ;
PATCHETT, AA ;
CHANG, RSL ;
LOTTI, VJ ;
CHEN, TB ;
SCHECK, SA ;
FAUST, KA ;
KIVLIGHN, SS ;
SCHORN, TS ;
ZINGARO, GJ ;
SIEGL, PKS .
JOURNAL OF MEDICINAL CHEMISTRY, 1993, 36 (21) :3207-3210
[4]
A facile synthesis of 2-amino-3H-quinazolin-4-ones with tandem Aza-Wittig reaction. [J].
Ding, MW ;
Zeng, GP ;
Wu, TJ .
SYNTHETIC COMMUNICATIONS, 2000, 30 (09) :1599-1604
[5]
ELSHIHI T, 1986, Z NATURFORSCH B, V41, P132
[6]
A general and efficient solid phase synthesis of quinazoline-2,4-diones [J].
Gordeev, MF ;
Hui, HC ;
Gordon, EM ;
Patel, DV .
TETRAHEDRON LETTERS, 1997, 38 (10) :1729-1732
[7]
Combinatorial chemistry of natural products: Solid phase synthesis of D- and L-cycloserine derivatives [J].
Gordeev, MF ;
Luehr, GW ;
Hui, HC ;
Gordon, EM ;
Patel, DV .
TETRAHEDRON, 1998, 54 (52) :15879-15890
[8]
Non-peptide glycoprotein IIb/IIIa antagonists .2. Design and in vivo evaluation of 3,4-dihydro-1(1H)-isoquinolinone-based antagonists and ethyl ester prodrugs [J].
Hutchinson, JH ;
Cook, JJ ;
Brashear, KM ;
Breslin, MJ ;
Glass, JD ;
Gould, RJ ;
Halczenko, W ;
Holahan, MA ;
Lynch, RJ ;
Sitko, GR ;
Stranieri, MT ;
Hartman, GD .
JOURNAL OF MEDICINAL CHEMISTRY, 1996, 39 (23) :4583-4591
[9]
Solid-phase synthesis of quinazolin-4(3H)-ones with three-point diversity [J].
Kesarwani, AP ;
Srivastava, GK ;
Rastogi, SK ;
Kundu, B .
TETRAHEDRON LETTERS, 2002, 43 (32) :5579-5581
[10]
Solid-phase synthesis of 2,3,5-triketopiperadine [J].
Makino, S ;
Nakanishi, E ;
Tsuji, T .
SYNLETT, 2003, (06) :817-820