Pyrazole-3(4)-carbaldehyde: synthesis, reactions and biological activity

被引：67

作者：

Abdel-Wahab, Bakr F. ^{[2
]}

Khidre, Rizk E. ^{[1
,3
]}

Farahat, Abdelbasset A. ^{[4
]}

机构：

[1] Gazan Univ, Fac Sci, Dept Chem, Gaza, Saudi Arabia

[2] King Abdulaziz Univ, Fac Sci & Arts, Dept Chem, Khulais Branch, Jeddah, Saudi Arabia

[3] Natl Res Ctr, Chem Ind Div, Giza 12622, Egypt

[4] Univ Mansoura, Fac Pharm, Dept Organ Pharmaceut Chem, Mansoura 35516, Egypt

来源：

ARKIVOC | 2011年

关键词：

Vilsmeier-Haack reaction; phenylhydrazone; pyrazolecarbaldehyde; chalcone; hydroxyalkylation; 4-FUNCTIONALLY SUBSTITUTED 3-HETERYLPYRAZOLES; ONE-POT SYNTHESIS; 2(3H)-FURANONES BEARING; ANTIMICROBIAL ACTIVITY; PYRAZOLE DERIVATIVES; DESIGN; 1,3-DIPHENYLPYRAZOLES; KETONES; CONDENSATION; FORMYLATION;

D O I：

10.3998/ark.5550190.0012.103

中图分类号：

O62 [有机化学];

学科分类号：

070303 [有机化学];

摘要：

This review deals with synthesis and reactions of pyrazole-3(4)-carbaldehydes as well as their biological activity. The data on the methods of synthesis, chemical reactions, and biological activity of these heterocycles published over the last years are reviewed here for the first time.

引用

页码：196 / 245

页数：50

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