Synthesis and aldose reductase inhibitory activity of benzoyl-amino acid derivatives

被引：7

作者：

Benvenuti, S ^{[1
]}

Severi, F ^{[1
]}

Costantino, L ^{[1
]}

Vampa, G ^{[1
]}

Melegari, M ^{[1
]}

机构：

[1] Univ Modena, Dipartimento Sci Farmaceut, I-41100 Modena, Italy

来源：

FARMACO | 1998年 / 53卷 / 06期

关键词：

benzoyl-L-amino acid derivatives; aldose reductase inhibitors;

D O I：

10.1016/S0014-827X(98)00038-X

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

A series of N-(4-methoxy, 4-fluoro, 4-trifluoromethyl and 4-nitrobenzoyl)-L-amino acids was synthesized and their inhibitory activity towards bovine lens aldose reductase (ALR2) was tested. (C) 1998 Elsevier Science S.A. AII rights reserved.

引用

页码：439 / 442

页数：4

共 13 条

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