Design, synthesis, and preclinical characterization of novel, highly selective indole estrogens

被引：122

作者：

Miller, CP

Collini, MD

Tran, BD

Harris, HA

Kharode, YP

Marzolf, JT

Moran, RA

Henderson, RA

Bender, RHW

Unwalla, RJ

Greenberger, LM

Yardley, JP

Abou-Gharbia, MA

Lyttle, CR

Komm, BS

机构：

[1] Wyeth Ayerst Res, Chem Sci, Radnor, PA 19087 USA

[2] Wyeth Ayerst Res, Womens Hlth Res Inst, Radnor, PA 19087 USA

[3] Wyeth Ayerst Res, Biol Chem, Radnor, PA 19087 USA

[4] Wyeth Ayerst Res, Oncol & Immunoinflammatory Res, Pearl River, NY 10965 USA

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 2001年 / 44卷 / 11期

关键词：

D O I：

10.1021/jm010086m

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1654 / 1657

页数：4

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