The synthesis of anthraquinone derivatives as potential anticancer agents

被引：16

作者：

Ge, P ^{[1
]}

Russell, RA ^{[1
]}

机构：

[1] DEAKIN UNIV,SCH BIOL & CHEM SCI,GEELONG,VIC 3217,AUSTRALIA

来源：

TETRAHEDRON | 1997年 / 53卷 / 51期

关键词：

D O I：

10.1016/S0040-4020(97)10195-8

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The simple anthracycline analogues 3a-c were synthesized as potential anticancer agents. Anodic oxidation of the phenol derivative 4, phthalide anion annelation of p-quinone monoacetals 5 and selective attachment of the side chain were the three key steps towards these target compounds. (C) 1997 Elsevier Science Ltd.

引用

页码：17469 / 17476

页数：8

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