6-chloro-5-methyl-1-[[2-[(2-methyl-3-pyridyl)oxy]-5-pyridyl]carbamoyl]-indoline (SB-242084): The first selective and brain penetrant 5-HT2C receptor antagonist

被引：78

作者：

Bromidge, SM

Duckworth, M

Forbes, IT

Ham, P

King, FD

Thewlis, KM

Blaney, FE

Naylor, CB

Blackburn, TP

Kennett, GA

Wood, MD

Clarke, SE

机构：

[1] SMITHKLINE BEECHAM PHARMACEUT CORP,DISCOVERY RES,DEPT NEUROSCI,HARLOW CM19 5AW,ESSEX,ENGLAND

[2] SMITHKLINE BEECHAM PHARMACEUT CORP,DISCOVERY RES,DEPT DRUG METAB & PHARMACOKINET,HARLOW CM19 5AW,ESSEX,ENGLAND

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1997年 / 40卷 / 22期

关键词：

D O I：

10.1021/jm970424c

中图分类号：

R914 [药物化学];

学科分类号：

100701 [药物化学];

摘要：

[No abstract available]

引用

页码：3494 / 3496

页数：3

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