Combinatorial synthesis of 2,9-substituted purines.

被引：86

作者：

Gray, NS ^{[1
]}

Kwon, S ^{[1
]}

Schultz, PG ^{[1
]}

机构：

[1] UNIV CALIF BERKELEY, DEPT CHEM, HOWARD HUGHES MED INST, BERKELEY, CA 94720 USA

来源：

TETRAHEDRON LETTERS | 1997年 / 38卷 / 07期

关键词：

D O I：

10.1016/S0040-4039(97)00014-2

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A method for the combinatorial synthesis of 2,9-substituted purines using a Mitsunobu reaction to alkylate the N-9 position and an amination reaction to install amines at the C-2 position has been developed. (C) 1997, Elsevier Science Ltd.

引用

页码：1161 / 1164

页数：4

共 7 条

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