(S)-(+)-4-[7-(2,2-dimethyl-1-oxopropoxy)-4-methyl-2-[4-[2-(1-piperidinyl)ethoxy]phenyl]-2H-1-benzopyran-3-yl]phenyl 2,2-dimethylpropanoate (EM-800): A highly potent, specific, and orally active nonsteroidal antiestrogen

被引：149

作者：

Gauthier, S

Caron, B

Cloutier, J

Dory, YL

Favre, A

Larouche, D

Mailhot, J

Ouellet, C

Schwerdtfeger, A

Leblanc, G

Martel, C

Simard, J

Merand, Y

Belanger, A

Labrie, C

Labrie, F

机构：

[1] CHU QUEBEC,CHUL,RES CTR,MOL ENDOCRINOL LAB,QUEBEC CITY,PQ G1V 4G2,CANADA

[2] UNIV LAVAL,QUEBEC CITY,PQ G1V 4G2,CANADA

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1997年 / 40卷 / 14期

关键词：

D O I：

10.1021/jm970095o

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：2117 / 2122

页数：6

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