New building blocks for peptide and depsipeptide modification N-glycosylated L-malic and L-citramalic acid derivatives

被引：7

作者：

Böttcher, C ^{[1
]}

Burger, K ^{[1
]}

机构：

[1] Univ Leipzig, Dept Organ Chem, D-04103 Leipzig, Germany

来源：

TETRAHEDRON LETTERS | 2002年 / 43卷 / 52期

关键词：

malic acid; citramalic acid; hexafluoroacetone; glycosyl amines; N-glycosylation; neoglycoconjugates;

D O I：

10.1016/S0040-4039(02)02285-2

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Neoglycoconjugates have been synthesized from L-malic acid/L-citramalic acid and beta-D-Ac(4)Glc-NH2/beta-D-Bzl(4)Glc-NH2 using hexafluoroacetone as protecting and activating agent. (C) 2002 Elsevier Science Ltd. All rights reserved.

引用

页码：9711 / 9714

页数：4

共 33 条

[1] Burger K, 1999, ANGEW CHEM INT EDIT, V38, P1414, DOI 10.1002/(SICI)1521-3773(19990517)38:10<1414::AID-ANIE1414>3.0.CO
[2] 2-L
[3] A new efficient approach to N-linked glycopeptoids
Burger, K
Böttcher, C
Radics, G
Hennig, L
[J]. TETRAHEDRON LETTERS, 2001, 42 (17) : 3061 - 3063
[4] NEW EFFICIENT STRATEGY FOR THE INCORPORATION OF (S)-ISOSERINE INTO PEPTIDES
BURGER, K
WINDEISEN, E
PIRES, R
[J]. JOURNAL OF ORGANIC CHEMISTRY, 1995, 60 (23) : 7641 - 7645
[5] BURGER K, 1999, ANGEW CHEM, V111, P1513
[6] Christiansen-Brams I, 1993, J CHEM SOC P1, V13, P1461
[7] DEGRADO WF, 1988, ADV PROTEIN CHEM, V39, P51
[8] PEPTIDE TO GLYCOPEPTIDE - GLYCOSYLATED OLIGOPEPTIDE RENIN INHIBITORS WITH ATTENUATED INVIVO CLEARANCE PROPERTIES
FISHER, JF
HARRISON, AW
BUNDY, GL
WILKINSON, KF
RUSH, BD
RUWART, MJ
[J]. JOURNAL OF MEDICINAL CHEMISTRY, 1991, 34 (10) : 3140 - 3143
[9] PEPTIDOMIMETICS FOR RECEPTOR LIGANDS DISCOVERY, DEVELOPMENT, AND MEDICAL PERSPECTIVES
GIANNIS, A
[J]. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 1993, 32 (09) : 1244 - 1267
[10] Giannis A., 1993, ANGEW CHEM, V105, P1303, DOI DOI 10.1002/ange.19931050905

← 1 2 3 4 →