Synthesis of radioiodinated aryl iodides via boronate precursors

被引：30

作者：

Kabalka, GW ^{[1
]}

Akula, MR

Zhang, JH

机构：

[1] Univ Tennessee, Dept Chem, Knoxville, TN 37966 USA

[2] Univ Tennessee, Dept Radiol, Knoxville, TN 37966 USA

来源：

NUCLEAR MEDICINE AND BIOLOGY | 2002年 / 29卷 / 08期

关键词：

arylboronates; chloramine-T; bis(neopentyl glycato)diboron; radiohalogenation;

D O I：

10.1016/S0969-8051(02)00344-X

中图分类号：

R8 [特种医学]; R445 [影像诊断学];

学科分类号：

1002 ; 100207 ; 1009 ;

摘要：

Arylboronate esters are converted to iodine-123 labeled aryl iodides using no-carrier-added iodine-123 labeled sodium iodide in the presence of chloramine-T. High yields of radiochemically pure products are obtained. (C) 2002 Elsevier Science Inc. All rights reserved.

引用

页码：841 / 843

页数：3

共 11 条

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