Synthesis of 2-aminoquinazoline-4(3H)-one derivatives as potential potassium channel openers

被引：10

作者：

Erb, B

Akue, R

Rigo, B

Pirotte, B

Couturier, D

机构：

[1] Ecole Hautes Etud Ind, Lab Engn Mol, F-59046 Lille, France

[2] Ctr Hosp Univ, Lab Chim Pharmaceut, B-4000 Liege, Belgium

[3] Univ Sci & Tech Lille Flandres Artois, Lab Engn Mol, F-59655 Villeneuve Dascq, France

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 2000年 / 37卷 / 02期

关键词：

D O I：

10.1002/jhet.5570370206

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Starting from 2-thioxoquinazolin-4-one, the synthesis of 2-amino-4(3H)-one derivatives, structurally related to potassium channels openers pinacidil and diazoxide, is described.

引用

页码：253 / 260

页数：8

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