A facile ligation approach to prepare three-helix bundles of HIV fusion-state protein mimetics

被引:25
作者
Tam, JP [1 ]
Yu, QT [1 ]
机构
[1] Vanderbilt Univ, Dept Microbiol & Immunol, Nashville, TN 37323 USA
关键词
D O I
10.1021/ol026932k
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
[GRAPHICS] We have designed a facile ligation approach to prepare three-helix bundles mimicking the HIV membrane fusion-state proteins that may be useful as inhibitors and vaccine candidates for blocking HIV infection.
引用
收藏
页码:4167 / 4170
页数:4
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