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Ras farnesyltransferase: A new therapeutic target
被引:250
作者
:
Leonard, DM
论文数:
0
引用数:
0
h-index:
0
机构:
Parke-Davis Pharmaceutical Research, Division of Warner-Lambert Company, Ann Arbor, MI 48105
Leonard, DM
机构
:
[1]
Parke-Davis Pharmaceutical Research, Division of Warner-Lambert Company, Ann Arbor, MI 48105
来源
:
JOURNAL OF MEDICINAL CHEMISTRY
|
1997年
/ 40卷
/ 19期
关键词
:
D O I
:
10.1021/jm970226l
中图分类号
:
R914 [药物化学];
学科分类号
:
100701 ;
摘要
:
[No abstract available]
引用
收藏
页码:2971 / 2990
页数:20
相关论文
共 185 条
[1]
Abrams SI, 1996, SEMIN ONCOL, V23, P118
[2]
ADAMSON P, 1992, J BIOL CHEM, V267, P20033
[3]
CLEAVAGE OF FARNESYLATED COOH-TERMINAL HEPTAPEPTIDE OF MOUSE N-RAS BY BRAIN MICROSOMAL-MEMBRANES - EVIDENCE FOR A CARBOXYPEPTIDASE, WHICH SPECIFICALLY REMOVES THE COOH-TERMINAL METHIONINE
AKOPYAN, TN
论文数:
0
引用数:
0
h-index:
0
机构:
UFR SCI PHARMACEUT & BIOL,DEPT CHIM ORGAN,CNRS,URA D1500,INSERM,UA498,U266,4 AVE OBSERV,F-75270 PARIS 06,FRANCE
UFR SCI PHARMACEUT & BIOL,DEPT CHIM ORGAN,CNRS,URA D1500,INSERM,UA498,U266,4 AVE OBSERV,F-75270 PARIS 06,FRANCE
AKOPYAN, TN
COUEDEL, Y
论文数:
0
引用数:
0
h-index:
0
机构:
UFR SCI PHARMACEUT & BIOL,DEPT CHIM ORGAN,CNRS,URA D1500,INSERM,UA498,U266,4 AVE OBSERV,F-75270 PARIS 06,FRANCE
UFR SCI PHARMACEUT & BIOL,DEPT CHIM ORGAN,CNRS,URA D1500,INSERM,UA498,U266,4 AVE OBSERV,F-75270 PARIS 06,FRANCE
COUEDEL, Y
BEAUMONT, A
论文数:
0
引用数:
0
h-index:
0
机构:
UFR SCI PHARMACEUT & BIOL,DEPT CHIM ORGAN,CNRS,URA D1500,INSERM,UA498,U266,4 AVE OBSERV,F-75270 PARIS 06,FRANCE
UFR SCI PHARMACEUT & BIOL,DEPT CHIM ORGAN,CNRS,URA D1500,INSERM,UA498,U266,4 AVE OBSERV,F-75270 PARIS 06,FRANCE
BEAUMONT, A
FOURNIEZALUSKI, MC
论文数:
0
引用数:
0
h-index:
0
机构:
UFR SCI PHARMACEUT & BIOL,DEPT CHIM ORGAN,CNRS,URA D1500,INSERM,UA498,U266,4 AVE OBSERV,F-75270 PARIS 06,FRANCE
UFR SCI PHARMACEUT & BIOL,DEPT CHIM ORGAN,CNRS,URA D1500,INSERM,UA498,U266,4 AVE OBSERV,F-75270 PARIS 06,FRANCE
FOURNIEZALUSKI, MC
ROQUES, BP
论文数:
0
引用数:
0
h-index:
0
机构:
UFR SCI PHARMACEUT & BIOL,DEPT CHIM ORGAN,CNRS,URA D1500,INSERM,UA498,U266,4 AVE OBSERV,F-75270 PARIS 06,FRANCE
UFR SCI PHARMACEUT & BIOL,DEPT CHIM ORGAN,CNRS,URA D1500,INSERM,UA498,U266,4 AVE OBSERV,F-75270 PARIS 06,FRANCE
ROQUES, BP
[J].
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS,
1992,
187
(03)
: 1336
-
1342
[4]
ANDEREGG RJ, 1988, J BIOL CHEM, V263, P18236
[5]
CAAX GERANYLGERANYL TRANSFERASE TRANSFERS FARNESYL AS EFFICIENTLY AS GERANYLGERANYL TO RHOB
ARMSTRONG, SA
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Molecular Genetics, Texas University SW Medical Center, Dallas
ARMSTRONG, SA
HANNAH, VC
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Molecular Genetics, Texas University SW Medical Center, Dallas
HANNAH, VC
GOLDSTEIN, JL
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Molecular Genetics, Texas University SW Medical Center, Dallas
GOLDSTEIN, JL
BROWN, MS
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Molecular Genetics, Texas University SW Medical Center, Dallas
BROWN, MS
[J].
JOURNAL OF BIOLOGICAL CHEMISTRY,
1995,
270
(14)
: 7864
-
7868
[6]
ENDOPROTEOLYTIC PROCESSING OF A FARNESYLATED PEPTIDE INVITRO
ASHBY, MN
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CALIF BERKELEY, DEPT MOLEC & CELL BIOL, DIV GENET, BERKELEY, CA 94720 USA
ASHBY, MN
KING, DS
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CALIF BERKELEY, DEPT MOLEC & CELL BIOL, DIV GENET, BERKELEY, CA 94720 USA
KING, DS
RINE, J
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CALIF BERKELEY, DEPT MOLEC & CELL BIOL, DIV GENET, BERKELEY, CA 94720 USA
RINE, J
[J].
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
1992,
89
(10)
: 4613
-
4617
[7]
RAS GENES
BARBACID, M
论文数:
0
引用数:
0
h-index:
0
BARBACID, M
[J].
ANNUAL REVIEW OF BIOCHEMISTRY,
1987,
56
: 779
-
827
[8]
INCORPORATION OF A PRODUCT OF MEVALONIC ACID METABOLISM INTO PROTEINS OF CHINESE-HAMSTER OVARY CELL-NUCLEI
BECK, LA
论文数:
0
引用数:
0
h-index:
0
BECK, LA
HOSICK, TJ
论文数:
0
引用数:
0
h-index:
0
HOSICK, TJ
SINENSKY, M
论文数:
0
引用数:
0
h-index:
0
SINENSKY, M
[J].
JOURNAL OF CELL BIOLOGY,
1988,
107
(04)
: 1307
-
1316
[9]
Bernhard EJ, 1996, CANCER RES, V56, P1727
[10]
RATIONAL DESIGN OF POTENT CARBOXYLIC-ACID BASED BISUBSTRATE INHIBITORS OF RAS FARNESYL-PROTEIN TRANSFERASE
BHIDE, RS
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol-Myers Squibb Pharmaceutical Research Institute, Princeton
BHIDE, RS
PATEL, DV
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol-Myers Squibb Pharmaceutical Research Institute, Princeton
PATEL, DV
PATEL, MM
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol-Myers Squibb Pharmaceutical Research Institute, Princeton
PATEL, MM
ROBINSON, SP
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol-Myers Squibb Pharmaceutical Research Institute, Princeton
ROBINSON, SP
HUNIHAN, LW
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol-Myers Squibb Pharmaceutical Research Institute, Princeton
HUNIHAN, LW
GORDON, EM
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol-Myers Squibb Pharmaceutical Research Institute, Princeton
GORDON, EM
[J].
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,
1994,
4
(17)
: 2107
-
2112
←
1
2
3
4
5
6
7
8
9
10
→
共 185 条
[1]
Abrams SI, 1996, SEMIN ONCOL, V23, P118
[2]
ADAMSON P, 1992, J BIOL CHEM, V267, P20033
[3]
CLEAVAGE OF FARNESYLATED COOH-TERMINAL HEPTAPEPTIDE OF MOUSE N-RAS BY BRAIN MICROSOMAL-MEMBRANES - EVIDENCE FOR A CARBOXYPEPTIDASE, WHICH SPECIFICALLY REMOVES THE COOH-TERMINAL METHIONINE
AKOPYAN, TN
论文数:
0
引用数:
0
h-index:
0
机构:
UFR SCI PHARMACEUT & BIOL,DEPT CHIM ORGAN,CNRS,URA D1500,INSERM,UA498,U266,4 AVE OBSERV,F-75270 PARIS 06,FRANCE
UFR SCI PHARMACEUT & BIOL,DEPT CHIM ORGAN,CNRS,URA D1500,INSERM,UA498,U266,4 AVE OBSERV,F-75270 PARIS 06,FRANCE
AKOPYAN, TN
COUEDEL, Y
论文数:
0
引用数:
0
h-index:
0
机构:
UFR SCI PHARMACEUT & BIOL,DEPT CHIM ORGAN,CNRS,URA D1500,INSERM,UA498,U266,4 AVE OBSERV,F-75270 PARIS 06,FRANCE
UFR SCI PHARMACEUT & BIOL,DEPT CHIM ORGAN,CNRS,URA D1500,INSERM,UA498,U266,4 AVE OBSERV,F-75270 PARIS 06,FRANCE
COUEDEL, Y
BEAUMONT, A
论文数:
0
引用数:
0
h-index:
0
机构:
UFR SCI PHARMACEUT & BIOL,DEPT CHIM ORGAN,CNRS,URA D1500,INSERM,UA498,U266,4 AVE OBSERV,F-75270 PARIS 06,FRANCE
UFR SCI PHARMACEUT & BIOL,DEPT CHIM ORGAN,CNRS,URA D1500,INSERM,UA498,U266,4 AVE OBSERV,F-75270 PARIS 06,FRANCE
BEAUMONT, A
FOURNIEZALUSKI, MC
论文数:
0
引用数:
0
h-index:
0
机构:
UFR SCI PHARMACEUT & BIOL,DEPT CHIM ORGAN,CNRS,URA D1500,INSERM,UA498,U266,4 AVE OBSERV,F-75270 PARIS 06,FRANCE
UFR SCI PHARMACEUT & BIOL,DEPT CHIM ORGAN,CNRS,URA D1500,INSERM,UA498,U266,4 AVE OBSERV,F-75270 PARIS 06,FRANCE
FOURNIEZALUSKI, MC
ROQUES, BP
论文数:
0
引用数:
0
h-index:
0
机构:
UFR SCI PHARMACEUT & BIOL,DEPT CHIM ORGAN,CNRS,URA D1500,INSERM,UA498,U266,4 AVE OBSERV,F-75270 PARIS 06,FRANCE
UFR SCI PHARMACEUT & BIOL,DEPT CHIM ORGAN,CNRS,URA D1500,INSERM,UA498,U266,4 AVE OBSERV,F-75270 PARIS 06,FRANCE
ROQUES, BP
[J].
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS,
1992,
187
(03)
: 1336
-
1342
[4]
ANDEREGG RJ, 1988, J BIOL CHEM, V263, P18236
[5]
CAAX GERANYLGERANYL TRANSFERASE TRANSFERS FARNESYL AS EFFICIENTLY AS GERANYLGERANYL TO RHOB
ARMSTRONG, SA
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Molecular Genetics, Texas University SW Medical Center, Dallas
ARMSTRONG, SA
HANNAH, VC
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Molecular Genetics, Texas University SW Medical Center, Dallas
HANNAH, VC
GOLDSTEIN, JL
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Molecular Genetics, Texas University SW Medical Center, Dallas
GOLDSTEIN, JL
BROWN, MS
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Molecular Genetics, Texas University SW Medical Center, Dallas
BROWN, MS
[J].
JOURNAL OF BIOLOGICAL CHEMISTRY,
1995,
270
(14)
: 7864
-
7868
[6]
ENDOPROTEOLYTIC PROCESSING OF A FARNESYLATED PEPTIDE INVITRO
ASHBY, MN
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CALIF BERKELEY, DEPT MOLEC & CELL BIOL, DIV GENET, BERKELEY, CA 94720 USA
ASHBY, MN
KING, DS
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CALIF BERKELEY, DEPT MOLEC & CELL BIOL, DIV GENET, BERKELEY, CA 94720 USA
KING, DS
RINE, J
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CALIF BERKELEY, DEPT MOLEC & CELL BIOL, DIV GENET, BERKELEY, CA 94720 USA
RINE, J
[J].
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
1992,
89
(10)
: 4613
-
4617
[7]
RAS GENES
BARBACID, M
论文数:
0
引用数:
0
h-index:
0
BARBACID, M
[J].
ANNUAL REVIEW OF BIOCHEMISTRY,
1987,
56
: 779
-
827
[8]
INCORPORATION OF A PRODUCT OF MEVALONIC ACID METABOLISM INTO PROTEINS OF CHINESE-HAMSTER OVARY CELL-NUCLEI
BECK, LA
论文数:
0
引用数:
0
h-index:
0
BECK, LA
HOSICK, TJ
论文数:
0
引用数:
0
h-index:
0
HOSICK, TJ
SINENSKY, M
论文数:
0
引用数:
0
h-index:
0
SINENSKY, M
[J].
JOURNAL OF CELL BIOLOGY,
1988,
107
(04)
: 1307
-
1316
[9]
Bernhard EJ, 1996, CANCER RES, V56, P1727
[10]
RATIONAL DESIGN OF POTENT CARBOXYLIC-ACID BASED BISUBSTRATE INHIBITORS OF RAS FARNESYL-PROTEIN TRANSFERASE
BHIDE, RS
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol-Myers Squibb Pharmaceutical Research Institute, Princeton
BHIDE, RS
PATEL, DV
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol-Myers Squibb Pharmaceutical Research Institute, Princeton
PATEL, DV
PATEL, MM
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol-Myers Squibb Pharmaceutical Research Institute, Princeton
PATEL, MM
ROBINSON, SP
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol-Myers Squibb Pharmaceutical Research Institute, Princeton
ROBINSON, SP
HUNIHAN, LW
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol-Myers Squibb Pharmaceutical Research Institute, Princeton
HUNIHAN, LW
GORDON, EM
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol-Myers Squibb Pharmaceutical Research Institute, Princeton
GORDON, EM
[J].
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,
1994,
4
(17)
: 2107
-
2112
←
1
2
3
4
5
6
7
8
9
10
→