Efficient synthesis of 1-substituted-5-hydroxymethylimidazole derivatives: Clean oxidative cleavage of 2-mercapto group

被引：14

作者：

Chang, JH ^{[1
]}

Lee, KW ^{[1
]}

Nam, DH ^{[1
]}

Kim, WS ^{[1
]}

Shin, K ^{[1
]}

机构：

[1] LGCI Ltd, Life Sci R&D, Taejon 305380, South Korea

来源：

ORGANIC PROCESS RESEARCH & DEVELOPMENT | 2002年 / 6卷 / 05期

关键词：

D O I：

10.1021/op020015c

中图分类号：

O69 [应用化学];

学科分类号：

081704 ;

摘要：

1-Substituted-5-hydroxymethylimidazoles were prepared through green desulfurization of their 2-mercapto derivatives by the treatment of 30% hydrogen peroxide in the presence of a catalytic amount of transition metal catalysts.

引用

页码：674 / 676

页数：3

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