Preparation and synthetic applications of sterically hindered secondary amines

被引：20

作者：

Kim, HO

Carroll, B

Lee, MS

机构：

[1] Molecumetics, Bellevue, WA 98005-2199

来源：

SYNTHETIC COMMUNICATIONS | 1997年 / 27卷 / 14期

关键词：

D O I：

10.1080/00397919708004114

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The preparation of sterically hindered secondary amino esters from the reaction of N-protected alpha-amino aldehydes and 3-, or Zero esters with alpha-amino esters by reductive amination is described. The resulting amino esters were converted to the beta-lactam or acylated to form N-acyl secondary amides.

引用

页码：2505 / 2515

页数：11

共 12 条

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