共 7 条
[1]
BLACKBURN BK, 1993, ANNU REP MED CHEM, V28, P79
[2]
Potent, orally active GPIIb/IIIa antagonists containing a nipecotic acid subunit. Structure-activity studies leading to the discovery of RWJ-53308
[J].
Hoekstra, WJ
;
Maryanoff, BE
;
Damiano, BP
;
Andrade-Gordon, P
;
Cohen, JH
;
Costanzo, MJ
;
Haertlein, BJ
;
Hecker, LR
;
Hulshizer, BL
;
Kauffman, JA
;
Keane, P
;
McComsey, DF
;
Mitchell, JA
;
Scott, L
;
Shah, RD
;
Yabut, SC
.
JOURNAL OF MEDICINAL CHEMISTRY,
1999, 42 (25)
:5254-5265

Hoekstra, WJ
论文数: 0 引用数: 0
h-index: 0
机构:
RW Johnson Pharmaceut Res Inst, Drug Discovery & New Prod Res, Spring House, PA 19477 USA RW Johnson Pharmaceut Res Inst, Drug Discovery & New Prod Res, Spring House, PA 19477 USA

Maryanoff, BE
论文数: 0 引用数: 0
h-index: 0
机构:
RW Johnson Pharmaceut Res Inst, Drug Discovery & New Prod Res, Spring House, PA 19477 USA RW Johnson Pharmaceut Res Inst, Drug Discovery & New Prod Res, Spring House, PA 19477 USA

Damiano, BP
论文数: 0 引用数: 0
h-index: 0
机构:
RW Johnson Pharmaceut Res Inst, Drug Discovery & New Prod Res, Spring House, PA 19477 USA RW Johnson Pharmaceut Res Inst, Drug Discovery & New Prod Res, Spring House, PA 19477 USA

Andrade-Gordon, P
论文数: 0 引用数: 0
h-index: 0
机构:
RW Johnson Pharmaceut Res Inst, Drug Discovery & New Prod Res, Spring House, PA 19477 USA RW Johnson Pharmaceut Res Inst, Drug Discovery & New Prod Res, Spring House, PA 19477 USA

Cohen, JH
论文数: 0 引用数: 0
h-index: 0
机构:
RW Johnson Pharmaceut Res Inst, Drug Discovery & New Prod Res, Spring House, PA 19477 USA RW Johnson Pharmaceut Res Inst, Drug Discovery & New Prod Res, Spring House, PA 19477 USA

Costanzo, MJ
论文数: 0 引用数: 0
h-index: 0
机构:
RW Johnson Pharmaceut Res Inst, Drug Discovery & New Prod Res, Spring House, PA 19477 USA RW Johnson Pharmaceut Res Inst, Drug Discovery & New Prod Res, Spring House, PA 19477 USA

Haertlein, BJ
论文数: 0 引用数: 0
h-index: 0
机构:
RW Johnson Pharmaceut Res Inst, Drug Discovery & New Prod Res, Spring House, PA 19477 USA RW Johnson Pharmaceut Res Inst, Drug Discovery & New Prod Res, Spring House, PA 19477 USA

Hecker, LR
论文数: 0 引用数: 0
h-index: 0
机构:
RW Johnson Pharmaceut Res Inst, Drug Discovery & New Prod Res, Spring House, PA 19477 USA RW Johnson Pharmaceut Res Inst, Drug Discovery & New Prod Res, Spring House, PA 19477 USA

Hulshizer, BL
论文数: 0 引用数: 0
h-index: 0
机构:
RW Johnson Pharmaceut Res Inst, Drug Discovery & New Prod Res, Spring House, PA 19477 USA RW Johnson Pharmaceut Res Inst, Drug Discovery & New Prod Res, Spring House, PA 19477 USA

Kauffman, JA
论文数: 0 引用数: 0
h-index: 0
机构:
RW Johnson Pharmaceut Res Inst, Drug Discovery & New Prod Res, Spring House, PA 19477 USA RW Johnson Pharmaceut Res Inst, Drug Discovery & New Prod Res, Spring House, PA 19477 USA

Keane, P
论文数: 0 引用数: 0
h-index: 0
机构:
RW Johnson Pharmaceut Res Inst, Drug Discovery & New Prod Res, Spring House, PA 19477 USA RW Johnson Pharmaceut Res Inst, Drug Discovery & New Prod Res, Spring House, PA 19477 USA

McComsey, DF
论文数: 0 引用数: 0
h-index: 0
机构:
RW Johnson Pharmaceut Res Inst, Drug Discovery & New Prod Res, Spring House, PA 19477 USA RW Johnson Pharmaceut Res Inst, Drug Discovery & New Prod Res, Spring House, PA 19477 USA

Mitchell, JA
论文数: 0 引用数: 0
h-index: 0
机构:
RW Johnson Pharmaceut Res Inst, Drug Discovery & New Prod Res, Spring House, PA 19477 USA RW Johnson Pharmaceut Res Inst, Drug Discovery & New Prod Res, Spring House, PA 19477 USA

Scott, L
论文数: 0 引用数: 0
h-index: 0
机构:
RW Johnson Pharmaceut Res Inst, Drug Discovery & New Prod Res, Spring House, PA 19477 USA RW Johnson Pharmaceut Res Inst, Drug Discovery & New Prod Res, Spring House, PA 19477 USA

Shah, RD
论文数: 0 引用数: 0
h-index: 0
机构:
RW Johnson Pharmaceut Res Inst, Drug Discovery & New Prod Res, Spring House, PA 19477 USA RW Johnson Pharmaceut Res Inst, Drug Discovery & New Prod Res, Spring House, PA 19477 USA

Yabut, SC
论文数: 0 引用数: 0
h-index: 0
机构:
RW Johnson Pharmaceut Res Inst, Drug Discovery & New Prod Res, Spring House, PA 19477 USA RW Johnson Pharmaceut Res Inst, Drug Discovery & New Prod Res, Spring House, PA 19477 USA
[3]
Conformational preferences in a benzodiazepine series of potent nonpeptide fibrinogen receptor antagonists
[J].
Keenan, RM
;
Callahan, JF
;
Samanen, JM
;
Bondinell, WE
;
Calvo, RR
;
Chen, LC
;
DeBrosse, C
;
Eggleston, DS
;
Haltiwanger, RC
;
Hwang, SM
;
Jakas, DR
;
Ku, TW
;
Miller, WH
;
Newlander, KA
;
Nichols, A
;
Parker, MF
;
Southhall, LS
;
Uzinskas, I
;
Vasko-Moser, JA
;
Venslavsky, JW
;
Wong, AS
;
Huffman, WF
.
JOURNAL OF MEDICINAL CHEMISTRY,
1999, 42 (04)
:545-559

Keenan, RM
论文数: 0 引用数: 0
h-index: 0
机构: SmithKline Beecham Pharmaceut, Div Res & Dev, Dept Med Chem, Collegeville, PA 19426 USA

Callahan, JF
论文数: 0 引用数: 0
h-index: 0
机构: SmithKline Beecham Pharmaceut, Div Res & Dev, Dept Med Chem, Collegeville, PA 19426 USA

Samanen, JM
论文数: 0 引用数: 0
h-index: 0
机构: SmithKline Beecham Pharmaceut, Div Res & Dev, Dept Med Chem, Collegeville, PA 19426 USA

Bondinell, WE
论文数: 0 引用数: 0
h-index: 0
机构: SmithKline Beecham Pharmaceut, Div Res & Dev, Dept Med Chem, Collegeville, PA 19426 USA

Calvo, RR
论文数: 0 引用数: 0
h-index: 0
机构: SmithKline Beecham Pharmaceut, Div Res & Dev, Dept Med Chem, Collegeville, PA 19426 USA

Chen, LC
论文数: 0 引用数: 0
h-index: 0
机构: SmithKline Beecham Pharmaceut, Div Res & Dev, Dept Med Chem, Collegeville, PA 19426 USA

DeBrosse, C
论文数: 0 引用数: 0
h-index: 0
机构: SmithKline Beecham Pharmaceut, Div Res & Dev, Dept Med Chem, Collegeville, PA 19426 USA

Eggleston, DS
论文数: 0 引用数: 0
h-index: 0
机构: SmithKline Beecham Pharmaceut, Div Res & Dev, Dept Med Chem, Collegeville, PA 19426 USA

Haltiwanger, RC
论文数: 0 引用数: 0
h-index: 0
机构: SmithKline Beecham Pharmaceut, Div Res & Dev, Dept Med Chem, Collegeville, PA 19426 USA

Hwang, SM
论文数: 0 引用数: 0
h-index: 0
机构: SmithKline Beecham Pharmaceut, Div Res & Dev, Dept Med Chem, Collegeville, PA 19426 USA

Jakas, DR
论文数: 0 引用数: 0
h-index: 0
机构: SmithKline Beecham Pharmaceut, Div Res & Dev, Dept Med Chem, Collegeville, PA 19426 USA

Ku, TW
论文数: 0 引用数: 0
h-index: 0
机构: SmithKline Beecham Pharmaceut, Div Res & Dev, Dept Med Chem, Collegeville, PA 19426 USA

Miller, WH
论文数: 0 引用数: 0
h-index: 0
机构: SmithKline Beecham Pharmaceut, Div Res & Dev, Dept Med Chem, Collegeville, PA 19426 USA

Newlander, KA
论文数: 0 引用数: 0
h-index: 0
机构: SmithKline Beecham Pharmaceut, Div Res & Dev, Dept Med Chem, Collegeville, PA 19426 USA

Nichols, A
论文数: 0 引用数: 0
h-index: 0
机构: SmithKline Beecham Pharmaceut, Div Res & Dev, Dept Med Chem, Collegeville, PA 19426 USA

Parker, MF
论文数: 0 引用数: 0
h-index: 0
机构: SmithKline Beecham Pharmaceut, Div Res & Dev, Dept Med Chem, Collegeville, PA 19426 USA

Southhall, LS
论文数: 0 引用数: 0
h-index: 0
机构: SmithKline Beecham Pharmaceut, Div Res & Dev, Dept Med Chem, Collegeville, PA 19426 USA

Uzinskas, I
论文数: 0 引用数: 0
h-index: 0
机构: SmithKline Beecham Pharmaceut, Div Res & Dev, Dept Med Chem, Collegeville, PA 19426 USA

Vasko-Moser, JA
论文数: 0 引用数: 0
h-index: 0
机构: SmithKline Beecham Pharmaceut, Div Res & Dev, Dept Med Chem, Collegeville, PA 19426 USA

Venslavsky, JW
论文数: 0 引用数: 0
h-index: 0
机构: SmithKline Beecham Pharmaceut, Div Res & Dev, Dept Med Chem, Collegeville, PA 19426 USA

Wong, AS
论文数: 0 引用数: 0
h-index: 0
机构: SmithKline Beecham Pharmaceut, Div Res & Dev, Dept Med Chem, Collegeville, PA 19426 USA

Huffman, WF
论文数: 0 引用数: 0
h-index: 0
机构: SmithKline Beecham Pharmaceut, Div Res & Dev, Dept Med Chem, Collegeville, PA 19426 USA
[4]
Tetrasubstituted imidazole inhibitors of cytokine release: Probing substituents in the N-1 position
[J].
Laufer, SA
;
Zimmermann, W
;
Ruff, KJ
.
JOURNAL OF MEDICINAL CHEMISTRY,
2004, 47 (25)
:6311-6325

Laufer, SA
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Tubingen, Inst Pharmaceut & Med Chem, Dept Pharm, D-72076 Tubingen, Germany Univ Tubingen, Inst Pharmaceut & Med Chem, Dept Pharm, D-72076 Tubingen, Germany

Zimmermann, W
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Tubingen, Inst Pharmaceut & Med Chem, Dept Pharm, D-72076 Tubingen, Germany Univ Tubingen, Inst Pharmaceut & Med Chem, Dept Pharm, D-72076 Tubingen, Germany

Ruff, KJ
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Tubingen, Inst Pharmaceut & Med Chem, Dept Pharm, D-72076 Tubingen, Germany Univ Tubingen, Inst Pharmaceut & Med Chem, Dept Pharm, D-72076 Tubingen, Germany
[5]
BREED: Generating novel inhibitors through hybridization of known ligands. Application to CDK2, P38, and HIV protease
[J].
Pierce, AC
;
Rao, G
;
Bemis, GW
.
JOURNAL OF MEDICINAL CHEMISTRY,
2004, 47 (11)
:2768-2775

Pierce, AC
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut, Cambridge, MA 02139 USA Vertex Pharmaceut, Cambridge, MA 02139 USA

Rao, G
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut, Cambridge, MA 02139 USA Vertex Pharmaceut, Cambridge, MA 02139 USA

Bemis, GW
论文数: 0 引用数: 0
h-index: 0
机构:
Vertex Pharmaceut, Cambridge, MA 02139 USA Vertex Pharmaceut, Cambridge, MA 02139 USA
[6]
Novel non-peptide fibrinogen receptor antagonists. 1. Synthesis and glycoprotein IIb-IIIa antagonistic activities of 1,3,4-trisubstituted 2-oxopiperazine derivatives incorporating side-chain functions of the RGDF peptide
[J].
Sugihara, H
;
Fukushi, H
;
Miyawaki, T
;
Imai, Y
;
Terashita, Z
;
Kawamura, M
;
Fujisawa, Y
;
Kita, S
.
JOURNAL OF MEDICINAL CHEMISTRY,
1998, 41 (04)
:489-502

Sugihara, H
论文数: 0 引用数: 0
h-index: 0
机构: Takeda Chem Ind Ltd, Div Pharmaceut Res, Yodogawa Ku, Osaka 5328686, Japan

Fukushi, H
论文数: 0 引用数: 0
h-index: 0
机构: Takeda Chem Ind Ltd, Div Pharmaceut Res, Yodogawa Ku, Osaka 5328686, Japan

Miyawaki, T
论文数: 0 引用数: 0
h-index: 0
机构: Takeda Chem Ind Ltd, Div Pharmaceut Res, Yodogawa Ku, Osaka 5328686, Japan

Imai, Y
论文数: 0 引用数: 0
h-index: 0
机构: Takeda Chem Ind Ltd, Div Pharmaceut Res, Yodogawa Ku, Osaka 5328686, Japan

Terashita, Z
论文数: 0 引用数: 0
h-index: 0
机构: Takeda Chem Ind Ltd, Div Pharmaceut Res, Yodogawa Ku, Osaka 5328686, Japan

Kawamura, M
论文数: 0 引用数: 0
h-index: 0
机构: Takeda Chem Ind Ltd, Div Pharmaceut Res, Yodogawa Ku, Osaka 5328686, Japan

Fujisawa, Y
论文数: 0 引用数: 0
h-index: 0
机构: Takeda Chem Ind Ltd, Div Pharmaceut Res, Yodogawa Ku, Osaka 5328686, Japan

Kita, S
论文数: 0 引用数: 0
h-index: 0
机构: Takeda Chem Ind Ltd, Div Pharmaceut Res, Yodogawa Ku, Osaka 5328686, Japan
[7]
Design and synthesis of 4-azaindoles as inhibitors of p38 MAP kinase
[J].
Trejo, A
;
Arzeno, H
;
Browner, M
;
Chanda, S
;
Cheng, S
;
Comer, DD
;
Dalrymple, SA
;
Dunten, P
;
Lafargue, J
;
Lovejoy, B
;
Freire-Moar, J
;
Lim, J
;
Mcintosh, J
;
Miller, J
;
Papp, E
;
Reuter, D
;
Roberts, R
;
Sanpablo, F
;
Saunders, J
;
Song, K
;
Villasenor, A
;
Warren, SD
;
Welch, M
;
Weller, P
;
Whiteley, PE
;
Zeng, L
;
Goldstein, DM
.
JOURNAL OF MEDICINAL CHEMISTRY,
2003, 46 (22)
:4702-4713

Trejo, A
论文数: 0 引用数: 0
h-index: 0
机构:
Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA

Arzeno, H
论文数: 0 引用数: 0
h-index: 0
机构:
Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA

Browner, M
论文数: 0 引用数: 0
h-index: 0
机构:
Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA

Chanda, S
论文数: 0 引用数: 0
h-index: 0
机构:
Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA

Cheng, S
论文数: 0 引用数: 0
h-index: 0
机构:
Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA

Comer, DD
论文数: 0 引用数: 0
h-index: 0
机构:
Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA

Dalrymple, SA
论文数: 0 引用数: 0
h-index: 0
机构:
Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA

Dunten, P
论文数: 0 引用数: 0
h-index: 0
机构:
Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA

Lafargue, J
论文数: 0 引用数: 0
h-index: 0
机构:
Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA

Lovejoy, B
论文数: 0 引用数: 0
h-index: 0
机构:
Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA

Freire-Moar, J
论文数: 0 引用数: 0
h-index: 0
机构:
Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA

Lim, J
论文数: 0 引用数: 0
h-index: 0
机构:
Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA

Mcintosh, J
论文数: 0 引用数: 0
h-index: 0
机构:
Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA

Miller, J
论文数: 0 引用数: 0
h-index: 0
机构:
Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA

Papp, E
论文数: 0 引用数: 0
h-index: 0
机构:
Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA

Reuter, D
论文数: 0 引用数: 0
h-index: 0
机构:
Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA

Roberts, R
论文数: 0 引用数: 0
h-index: 0
机构:
Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA

Sanpablo, F
论文数: 0 引用数: 0
h-index: 0
机构:
Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA

Saunders, J
论文数: 0 引用数: 0
h-index: 0
机构:
Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA

Song, K
论文数: 0 引用数: 0
h-index: 0
机构:
Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA

Villasenor, A
论文数: 0 引用数: 0
h-index: 0
机构:
Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA

Warren, SD
论文数: 0 引用数: 0
h-index: 0
机构:
Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA

Welch, M
论文数: 0 引用数: 0
h-index: 0
机构:
Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA

Weller, P
论文数: 0 引用数: 0
h-index: 0
机构:
Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA

Whiteley, PE
论文数: 0 引用数: 0
h-index: 0
机构:
Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA

Zeng, L
论文数: 0 引用数: 0
h-index: 0
机构:
Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA

Goldstein, DM
论文数: 0 引用数: 0
h-index: 0
机构:
Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Dept Med Chem, Palo Alto, CA 94304 USA