One pot biaryl synthesis via in situ boronate formation

被引：112

作者：

Giroux, A

Han, YX

Prasit, P

机构：

[1] Department of Medicinal Chemistry, Merck-Frosst Ctr. Therapeut. Res., Pointe-Claire-Dorval, Que. H9R 4P8

来源：

TETRAHEDRON LETTERS | 1997年 / 38卷 / 22期

关键词：

D O I：

10.1016/S0040-4039(97)00767-3

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The palladium-catalyzed cross-coupling reaction of aryl halides or aryl triflates with diborane 1 yielded structurally diverse aryl boronates which were reacted in situ with aryl halides or aryl triflates to afford a variety of biaryls in moderate to high yield. (C) 1997 Elsevier Science Ltd.

引用

页码：3841 / 3844

页数：4

共 29 条

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