Copper-catalyzed amination of aryl halides: single-step synthesis of triarylamines

被引：155

作者：

Kelkar, AA ^{[1
]}

Patil, NM ^{[1
]}

Chaudhari, RV ^{[1
]}

机构：

[1] Natl Chem Lab, Homogeneous Catalysis Div, Pune 411008, Maharashtra, India

来源：

TETRAHEDRON LETTERS | 2002年 / 43卷 / 40期

关键词：

D O I：

10.1016/S0040-4039(02)01708-2

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A simple and efficient methodology for the synthesis of triarylamines in a single step has been demonstrated using a ligand-free CuI catalyst and potassium tertiary butoxide as the base. Use of chelating ligands leads to the formation of triarylamine derivatives selectively (95% yield) with high catalytic activity. (C) 2002 Published by Elsevier Science Ltd.

引用

页码：7143 / 7146

页数：4

共 19 条

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