Synthesis and fungicidal activities of 4H-imidazolin-4-ones containing sulfur substituent

被引：23

作者：

Ding, MW ^{[1
]}

Zeng, GP ^{[1
]}

Liu, ZJ ^{[1
]}

机构：

[1] Cent China Normal Univ, Inst Organ Synth, Wuhan 430079, Peoples R China

来源：

PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS | 2002年 / 177卷 / 05期

基金：

中国国家自然科学基金;

关键词：

Aza-Wittig reaction; fungicidal activities; 4H-imidazolin-4-ones; synthesis;

D O I：

10.1080/10426500211728

中图分类号：

O61 [无机化学];

学科分类号：

070301 ; 081704 ;

摘要：

4H-Imidazolin-4-ones 3 and 4 were synthesized respectively by base catalytic reactions of 4-methylthiophenol or phenthiol with carbodiimides 2, which were obtained via aza-Wittig reaction of iminophosphorane 1 with aromatic isocyanates. 3 and 4 exhibited good fungicidal activity against Pellicularia sasakii.

引用

页码：1315 / 1321

页数：7

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