共 12 条
Molecules, Materials, Medicines (M3): Linking Molecules to Medicines through Pharmaceutical Material Science
被引:13
作者:

Almarsson, Oern
论文数: 0 引用数: 0
h-index: 0
机构:
Moderna Therapeut Inc, Cambridge, MA 02139 USA Moderna Therapeut Inc, Cambridge, MA 02139 USA

Vadas, Elizabeth B.
论文数: 0 引用数: 0
h-index: 0
机构:
InSciTech Inc, Dorval, PQ, Canada Moderna Therapeut Inc, Cambridge, MA 02139 USA
机构:
[1] Moderna Therapeut Inc, Cambridge, MA 02139 USA
[2] InSciTech Inc, Dorval, PQ, Canada
关键词:
D O I:
10.1021/acs.cgd.5b01417
中图分类号:
O6 [化学];
学科分类号:
0703 ;
摘要:
[No abstract available]
引用
收藏
页码:5645 / 5647
页数:3
相关论文
共 12 条
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Crystal engineering of the composition of pharmaceutical phases.: Do pharmaceutical co-crystals represent a new path to improved medicines?
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Almarsson, Ö
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Zaworotko, MJ
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Bak, Annette
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Amgen Inc, Dept Pharmaceut, Cambridge, MA 02139 USA Amgen Inc, Dept Pharmaceut, Cambridge, MA 02139 USA

Gore, Anu
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h-index: 0
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Amgen Inc, Dept Pharmaceut, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Pharmaceut, Cambridge, MA 02139 USA

Yanez, Evelyn
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h-index: 0
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Amgen Inc, Dept Pharmaceut, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Pharmaceut, Cambridge, MA 02139 USA

Stanton, Mary
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Amgen Inc, Dept Pharmaceut, Cambridge, MA 02139 USA Amgen Inc, Dept Pharmaceut, Cambridge, MA 02139 USA

Tufekcic, Sunita
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h-index: 0
机构:
Amgen Inc, Dept Pharmaceut, Cambridge, MA 02139 USA Amgen Inc, Dept Pharmaceut, Cambridge, MA 02139 USA

Syed, Rashid
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h-index: 0
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Amgen Inc, Mol Struct, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Pharmaceut, Cambridge, MA 02139 USA

Akrami, Anna
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h-index: 0
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Amgen Inc, Pharmacokinet & Drug Metab, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Pharmaceut, Cambridge, MA 02139 USA

Rose, Mark
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h-index: 0
机构:
Amgen Inc, Pharmacokinet & Drug Metab, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Pharmaceut, Cambridge, MA 02139 USA

Surapaneni, Sekhar
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h-index: 0
机构:
Amgen Inc, Pharmacokinet & Drug Metab, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Pharmaceut, Cambridge, MA 02139 USA

Bostick, Tracy
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h-index: 0
机构:
Amgen Inc, Chem Res & Dev, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Pharmaceut, Cambridge, MA 02139 USA

King, Anthony
论文数: 0 引用数: 0
h-index: 0
机构:
Amgen Inc, Chem Res & Dev, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Pharmaceut, Cambridge, MA 02139 USA

Neervannan, Sesha
论文数: 0 引用数: 0
h-index: 0
机构:
Amgen Inc, Dept Pharmaceut, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Pharmaceut, Cambridge, MA 02139 USA

Ostovic, Drazen
论文数: 0 引用数: 0
h-index: 0
机构:
Amgen Inc, Dept Pharmaceut, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Pharmaceut, Cambridge, MA 02139 USA

Koparkar, Arun
论文数: 0 引用数: 0
h-index: 0
机构:
Amgen Inc, Dept Pharmaceut, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Pharmaceut, Cambridge, MA 02139 USA
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Development of an Early-Phase Bulk Enabling Route to Sodium-Dependent Glucose Cotransporter 2 Inhibitor Ertugliflozin
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Lehner, Richard S.
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ORGANIC PROCESS RESEARCH & DEVELOPMENT,
2014, 18 (01)
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Bernhardson, David
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res & Dev, Med Chem, Groton, CT 06340 USA Pfizer Worldwide Res & Dev, Chem Res & Dev, Groton, CT 06340 USA

Brandt, Thomas A.
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res & Dev, Chem Res & Dev, Groton, CT 06340 USA Pfizer Worldwide Res & Dev, Chem Res & Dev, Groton, CT 06340 USA

Hulford, Catherine A.
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h-index: 0
机构:
Pfizer Worldwide Res & Dev, Med Chem, Groton, CT 06340 USA Pfizer Worldwide Res & Dev, Chem Res & Dev, Groton, CT 06340 USA

Lehner, Richard S.
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h-index: 0
机构:
Pfizer Worldwide Res & Dev, Chem Res & Dev, Groton, CT 06340 USA Pfizer Worldwide Res & Dev, Chem Res & Dev, Groton, CT 06340 USA

Preston, Brian R.
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h-index: 0
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Pfizer Worldwide Res & Dev, Res Analyt, Groton, CT 06340 USA Pfizer Worldwide Res & Dev, Chem Res & Dev, Groton, CT 06340 USA

Price, Kristin
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h-index: 0
机构:
Pfizer Worldwide Res & Dev, Chem Res & Dev, Groton, CT 06340 USA Pfizer Worldwide Res & Dev, Chem Res & Dev, Groton, CT 06340 USA

Sagal, John F.
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h-index: 0
机构:
Pfizer Worldwide Res & Dev, Chem Res & Dev, Groton, CT 06340 USA Pfizer Worldwide Res & Dev, Chem Res & Dev, Groton, CT 06340 USA

St Pierre, Michael J.
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res & Dev, Chem Res & Dev, Groton, CT 06340 USA Pfizer Worldwide Res & Dev, Chem Res & Dev, Groton, CT 06340 USA

Thompson, Peter H.
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res & Dev, Chem Res & Dev, Groton, CT 06340 USA Pfizer Worldwide Res & Dev, Chem Res & Dev, Groton, CT 06340 USA

Thuma, Benjamin
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Worldwide Res & Dev, Med Chem, Groton, CT 06340 USA Pfizer Worldwide Res & Dev, Chem Res & Dev, Groton, CT 06340 USA
[4]
Assessment of the physical stability of lyophilized MK-0591 by differential scanning calorimetry
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Clas, SD
论文数: 0 引用数: 0
h-index: 0
机构:
UNIV WISCONSIN,SCH PHARM,MADISON,WI 53706 UNIV WISCONSIN,SCH PHARM,MADISON,WI 53706

Cotton, M
论文数: 0 引用数: 0
h-index: 0
机构:
UNIV WISCONSIN,SCH PHARM,MADISON,WI 53706 UNIV WISCONSIN,SCH PHARM,MADISON,WI 53706

Moran, E
论文数: 0 引用数: 0
h-index: 0
机构:
UNIV WISCONSIN,SCH PHARM,MADISON,WI 53706 UNIV WISCONSIN,SCH PHARM,MADISON,WI 53706

Spagnoli, S
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h-index: 0
机构:
UNIV WISCONSIN,SCH PHARM,MADISON,WI 53706 UNIV WISCONSIN,SCH PHARM,MADISON,WI 53706

Zografi, G
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h-index: 0
机构:
UNIV WISCONSIN,SCH PHARM,MADISON,WI 53706 UNIV WISCONSIN,SCH PHARM,MADISON,WI 53706

Vadas, EB
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Connelly, Patrick R.
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Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USA

Snyder, Phillip W.
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Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USA

Zhang, Yuegang
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机构:
Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USA

McClain, Brian
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机构:
Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USA

Quinn, Brian P.
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h-index: 0
机构:
Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USA

Johnston, Steve
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h-index: 0
机构:
Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USA

Medek, Ales
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h-index: 0
机构:
Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USA

Tanoury, Jerry
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机构:
Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USA

Griffith, James
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机构:
Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USA

Walters, W. Patrick
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h-index: 0
机构:
Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USA

Dokou, Eleni
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h-index: 0
机构:
Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USA

Knezic, Dragutin
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h-index: 0
机构:
Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USA

Bransford, Philip
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Demuth, B.
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Budapest Univ Technol & Econ, Dept Organ Chem & Technol, H-1111 Budapest, Hungary Budapest Univ Technol & Econ, Dept Organ Chem & Technol, H-1111 Budapest, Hungary

Nagy, Z. K.
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h-index: 0
机构:
Budapest Univ Technol & Econ, Dept Organ Chem & Technol, H-1111 Budapest, Hungary Budapest Univ Technol & Econ, Dept Organ Chem & Technol, H-1111 Budapest, Hungary

Balogh, A.
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h-index: 0
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Budapest Univ Technol & Econ, Dept Organ Chem & Technol, H-1111 Budapest, Hungary Budapest Univ Technol & Econ, Dept Organ Chem & Technol, H-1111 Budapest, Hungary

Vigh, T.
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Budapest Univ Technol & Econ, Dept Organ Chem & Technol, H-1111 Budapest, Hungary Budapest Univ Technol & Econ, Dept Organ Chem & Technol, H-1111 Budapest, Hungary

Marosi, G.
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h-index: 0
机构:
Budapest Univ Technol & Econ, Dept Organ Chem & Technol, H-1111 Budapest, Hungary Budapest Univ Technol & Econ, Dept Organ Chem & Technol, H-1111 Budapest, Hungary

Verreck, G.
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h-index: 0
机构:
Johnson & Johnson, Div Janssen Pharmaceut, Pharmaceut Res & Dev, B-2340 Beerse, Belgium Budapest Univ Technol & Econ, Dept Organ Chem & Technol, H-1111 Budapest, Hungary

Van Assche, I.
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h-index: 0
机构:
Johnson & Johnson, Div Janssen Pharmaceut, Pharmaceut Res & Dev, B-2340 Beerse, Belgium Budapest Univ Technol & Econ, Dept Organ Chem & Technol, H-1111 Budapest, Hungary

Brewster, M. E.
论文数: 0 引用数: 0
h-index: 0
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Johnson & Johnson, Div Janssen Pharmaceut, Pharmaceut Res & Dev, B-2340 Beerse, Belgium Budapest Univ Technol & Econ, Dept Organ Chem & Technol, H-1111 Budapest, Hungary
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Loftsson, Thorsteinn
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h-index: 0
机构:
Univ Iceland, Fac Pharmaceut Sci, IS-107 Reykjavik, Iceland Univ Iceland, Fac Pharmaceut Sci, IS-107 Reykjavik, Iceland

Brewster, Marcus E.
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h-index: 0
机构:
Johnson & Johnson, Janssen Res & Dev, Pharmaceut Dev & Mfg Sci, B-2340 Beerse, Belgium Univ Iceland, Fac Pharmaceut Sci, IS-107 Reykjavik, Iceland
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On the importance of synthetic organic chemistry in drug discovery: reflections on the discovery of antidiabetic agent ertugliflozin
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Mascitti, Vincent
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Mascitti, Vincent
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机构:
Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA

Thuma, Benjamin A.
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h-index: 0
机构:
Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA

Smith, Aaron C.
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h-index: 0
机构:
Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA

Robinson, Ralph P.
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h-index: 0
机构:
Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA

Brandt, Thomas
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA

Kalgutkar, Amit S.
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h-index: 0
机构:
Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA

Maurer, Tristan S.
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h-index: 0
机构:
Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA

Samas, Brian
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h-index: 0
机构:
Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA

Sharma, Raman
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h-index: 0
机构:
Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA
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Mosquera-Giraldo, Laura I.
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Purdue Univ, Coll Pharm, Dept Ind & Phys Pharm, W Lafayette, IN 47907 USA Purdue Univ, Coll Pharm, Dept Ind & Phys Pharm, W Lafayette, IN 47907 USA

Taylor, Lynne S.
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Newman, Ann
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Seventh St Dev Grp, Lafayette, IN 47901 USA Seventh St Dev Grp, Lafayette, IN 47901 USA

Knipp, Gregory
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h-index: 0
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Purdue Univ, Dept Ind & Phys Pharm, Sch Pharm, W Lafayette, IN 47907 USA Seventh St Dev Grp, Lafayette, IN 47901 USA

Zografi, George
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Wisconsin Madison, Sch Pharm, Madison, WI 53705 USA Seventh St Dev Grp, Lafayette, IN 47901 USA