Palladium-catalysed α-arylation of esters and amides under microwave conditions

被引：36

作者：

Bentz, E

Moloney, MG

Westaway, SM

机构：

[1] Univ Oxford, Dept Chem, Cent Res Lab, Oxford OX1 3TA, England

[2] GlaxoSmithKline Res Ltd, Dept Med Chem Neurol, Harlow CM19 5AW, Essex, England

[3] GlaxoSmithKline Res Ltd, GI CEDD, Harlow CM19 5AW, Essex, England

来源：

TETRAHEDRON LETTERS | 2004年 / 45卷 / 40期

基金：

英国工程与自然科学研究理事会;

关键词：

arylation; Reformatsky; catalysis; microwave;

D O I：

10.1016/j.tetlet.2004.08.074

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A rapid and convenient approach for the alpha-arylation of esters and amides using Reformatsky reagents under a microwave accelerated reaction protocol has been established. (C) 2004 Elsevier Ltd. All rights reserved.

引用

页码：7395 / 7397

页数：3

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