Chloromethyl sulfones from sulfonyl chlorides via a one-pot procedure

被引：30

作者：

Antane, S ^{[1
]}

Bernotas, R ^{[1
]}

Li, YF ^{[1
]}

McDevitt, R ^{[1
]}

Yan, YF ^{[1
]}

机构：

[1] Wyeth Res, Chen & Screening Sci, Princeton, NJ 08543 USA

来源：

SYNTHETIC COMMUNICATIONS | 2004年 / 34卷 / 13期

关键词：

chloromethyl sulfones; one-pot procedure; sulfinate salts; sulfonyl chlorides;

D O I：

10.1081/SCC-120039498

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A simplified one-pot transformation of a diverse set of aryl- and heteroaryl-sulfonyl chlorides into the corresponding chloromethyl sulfones is described.

引用

页码：2443 / 2449

页数：7

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