Condensation reactions of a nitrodienamine with Grignard and organocopper reagents prepared from indole derivatives

被引：13

作者：

Koike, T ^{[1
]}

Takeuchi, N ^{[1
]}

Hagiwara, M ^{[1
]}

Yamazaki, K ^{[1
]}

Tobinaga, S ^{[1
]}

机构：

[1] Showa Coll Pharmaceut Sci, Tokyo 1948543, Japan

来源：

HETEROCYCLES | 1999年 / 51卷 / 11期

关键词：

D O I：

10.3987/COM-99-8684

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Condensation reactions of a nitrodienamine (1) with Grignard and organocopper reagents prepared from indole derivatives were investigated. Indolyl Grignard reagents were prepared from 4-bromoindole (3a), 5-bromoindole (3b), 6-bromoindole (3c), and 5-nitroindole (3d) using methylmagnesium bromide. Indolyl organocopper reagents were prepared from indole (3e), 2-methylindole (3f), and 3-methylindole (3g) using dimethylcopperlithium.

引用

页码：2687 / 2695

页数：9

共 14 条

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