The synthetic pentasaccharide fondaparinux sodium does not interact with oral warfarin

被引:13
作者
Faaij, RA
Burggraaf, J
Schoemaker, RC
de Greef, R
Cohen, AF
机构
[1] Ctr Human Drug Res, CHDR, NL-2333 CL Leiden, Netherlands
[2] NV Organon, Oss, Netherlands
关键词
D O I
10.2165/00003088-200241002-00004
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
[No abstract available]
引用
收藏
页码:27 / 29
页数:3
相关论文
共 11 条
[1]  
BIGGS R, 1972, HUMAN BLOOD COAGULAT
[2]   PHARMACOKINETIC AND ANTITHROMBOTIC PROPERTIES OF 2 PENTASACCHARIDES WITH HIGH-AFFINITY TO ANTITHROMBIN-III IN THE RABBIT - COMPARISON WITH CY216 [J].
CARRIE, D ;
CARANOBE, C ;
SAIVIN, S ;
HOUIN, G ;
PETITOU, M ;
LORMEAU, JC ;
VANBOECKEL, C ;
MEULEMAN, D ;
BONEU, B .
BLOOD, 1994, 84 (08) :2571-2577
[3]   The effect of warfarin on the pharmacokinetics and pharmacodynamics of napsagatran in healthy male volunteers [J].
Faaij, RA ;
van Griensven, JMT ;
Schoemaker, RC ;
Goggin, T ;
Guenzi, A ;
Kroon, JM ;
Burggraaf, J ;
Cohen, AF .
EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY, 2001, 57 (01) :25-29
[4]  
HOBBELEN PMJ, 1990, THROMB HAEMOSTASIS, V63, P265
[5]   Fondaparinux sodium is not metabolised in mammalian liver fractions and does not inhibit cytochrome P450-mediated metabolism of concomitant drugs [J].
Lieu, C ;
Shi, JA ;
Donat, F ;
Van Horn, R ;
Brian, W ;
Newton, J ;
Delbressine, L ;
Vos, R .
CLINICAL PHARMACOKINETICS, 2002, 41 (Suppl 2) :19-26
[6]   Fondaparinux sodium mechanism of action -: Identification of specific binding to purified and human plasma-derived proteins [J].
Paolucci, F ;
Claviés, MC ;
Donat, F ;
Necciari, J .
CLINICAL PHARMACOKINETICS, 2002, 41 (Suppl 2) :11-18
[7]   MECHANISM OF ANTITHROMBIN-III INHIBITION OF FACTOR VIIA TISSUE FACTOR ACTIVITY ON CELL-SURFACES - COMPARISON WITH TISSUE FACTOR PATHWAY INHIBITOR FACTOR XA-INDUCED INHIBITION OF FACTOR VIIA TISSUE FACTOR ACTIVITY [J].
RAO, LVM ;
NORDFANG, O ;
HOANG, AD ;
PENDURTHI, UR .
BLOOD, 1995, 85 (01) :121-129
[8]   COMPARATIVE EFFECTS OF RANITIDINE AND CIMETIDINE ON THE PHARMACOKINETICS AND PHARMACODYNAMICS OF WARFARIN IN MAN [J].
TOON, S ;
HOPKINS, KJ ;
GARSTANG, FM ;
ROWLAND, M .
EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY, 1987, 32 (02) :165-172
[9]   ENOXACIN-WARFARIN INTERACTION - PHARMACOKINETIC AND STEREOCHEMICAL ASPECTS [J].
TOON, S ;
HOPKINS, KJ ;
GARSTANG, FM ;
AARONS, L ;
SEDMAN, A ;
ROWLAND, M .
CLINICAL PHARMACOLOGY & THERAPEUTICS, 1987, 42 (01) :33-41
[10]   INVESTIGATIONS INTO THE POTENTIAL EFFECTS OF MULTIPLE DOSE KETOROLAC ON THE PHARMACOKINETICS AND PHARMACODYNAMICS OF RACEMIC WARFARIN [J].
TOON, S ;
HOLT, BL ;
MULLINS, FGP ;
BULLINGHAM, R ;
AARONS, L ;
ROWLAND, M .
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1990, 30 (05) :743-750