New targets for therapeutic attack

被引:9
作者
Wakeling, AE
Barker, AJ
Davies, DH
Brown, DS
Green, LR
Cartlidge, SA
Woodburn, JR
机构
关键词
D O I
10.1677/erc.0.0040351
中图分类号
R73 [肿瘤学];
学科分类号
100214 ;
摘要
引用
收藏
页码:351 / 355
页数:5
相关论文
共 18 条
[1]  
BARKER AJ, 1992, Patent No. 520722
[2]   4,5-DIANILINOPHTHALIMIDE - A PROTEIN-TYROSINE KINASE INHIBITOR WITH SELECTIVITY FOR THE EPIDERMAL GROWTH-FACTOR RECEPTOR SIGNAL-TRANSDUCTION PATHWAY AND POTENT IN-VIVO ANTITUMOR-ACTIVITY [J].
BUCHDUNGER, E ;
TRINKS, U ;
METT, H ;
REGENASS, U ;
MULLER, M ;
MEYER, T ;
MCGLYNN, E ;
PINNA, LA ;
TRAXLER, P ;
LYDON, NB .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1994, 91 (06) :2334-2338
[3]  
BURKE T R JR, 1992, Drugs of the Future, V17, P119
[4]   THE EGF RECEPTOR SYSTEM AS A TARGET FOR ANTITUMOR THERAPY [J].
ENNIS, BW ;
LIPPMAN, ME ;
DICKSON, RB .
CANCER INVESTIGATION, 1991, 9 (05) :553-562
[5]   A SPECIFIC INHIBITOR OF THE EPIDERMAL GROWTH-FACTOR RECEPTOR TYROSINE KINASE [J].
FRY, DW ;
KRAKER, AJ ;
MCMICHAEL, A ;
AMBROSO, LA ;
NELSON, JM ;
LEOPOLD, WR ;
CONNERS, RW ;
BRIDGES, AJ .
SCIENCE, 1994, 265 (5175) :1093-1095
[6]   PHARMACEUTICAL RESEARCH IN MOLECULAR ONCOLOGY [J].
GIBBS, JB ;
OLIFF, A .
CELL, 1994, 79 (02) :193-198
[7]   PREVALENCE OF ABERRANT EXPRESSION OF THE EPIDERMAL GROWTH-FACTOR RECEPTOR IN HUMAN CANCERS [J].
GULLICK, WJ .
BRITISH MEDICAL BULLETIN, 1991, 47 (01) :87-98
[8]   Eukaryotic protein kinases [J].
Hanks, Steven K. .
CURRENT OPINION IN STRUCTURAL BIOLOGY, 1991, 1 (03) :369-383
[9]   SH2 AND SH3 DOMAINS - ELEMENTS THAT CONTROL INTERACTIONS OF CYTOPLASMIC SIGNALING PROTEINS [J].
KOCH, CA ;
ANDERSON, D ;
MORAN, MF ;
ELLIS, C ;
PAWSON, T .
SCIENCE, 1991, 252 (5006) :668-674
[10]  
POWIS G, 1994, ANTI-CANCER DRUG DES, V9, P263