Improved synthesis of pyrrolo[1,2-c]pyrimidine and derivatives

被引：24

作者：

Minguez, JM ^{[1
]}

Vaquero, JJ ^{[1
]}

GarciaNavio, JL ^{[1
]}

AlvarezBuilla, J ^{[1
]}

机构：

[1] UNIV ALCALA DE HENARES, DEPT QUIM ORGAN, E-28871 ALCALA DE HENARES, SPAIN

来源：

TETRAHEDRON LETTERS | 1996年 / 37卷 / 24期

关键词：

D O I：

10.1016/0040-4039(96)00812-X

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

An improved synthesis of pyrrolo[1,2-c]pyrimidine derivatives by cyclocondensation of pyrrole-2-carboxaldehydes with tosylmethyl isocyanide followed by desulfonylation of the resulting 2-tosylpyrrolo[1,2-c]pyrimidines with sodium amalgam is described Copyright (C) 1996 Elsevier Science Ltd

引用

页码：4263 / 4266

页数：4

共 15 条

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