Discovering drugs through biological transformation: Role of pharmacologically active metabolites in drug discovery

被引：97

作者：

Fura, A

Shu, YZ

Zhu, MS

Hanson, RL

Roongta, V

Humphreys, WG

机构：

[1] Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08534 USA

[2] Bristol Myers Squibb Co, Pharmaceut Res Inst, Wallingford, CT 06492 USA

[3] Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA

[4] Bristol Myers Squibb Co, Pharmaceut Res Inst, New Brunswick, NJ 08903 USA

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 2004年 / 47卷 / 18期

关键词：

D O I：

10.1021/jm040066v

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

[No abstract available]

引用

页码：4339 / 4351

页数：13

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