Solid phase synthesis of tetrahydroisoquinolines & tetrahydroimidazopyridines

被引：43

作者：

Hutchins, SM

Chapman, KT

机构：

[1] Automated Synthesis Group, Dept. of Molec. Design and Diversity, Merck Research Laboratories, Rahway

来源：

TETRAHEDRON LETTERS | 1996年 / 37卷 / 28期

关键词：

D O I：

10.1016/0040-4039(96)00996-3

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The preparation of 1,2,3,4-tetrahydroisoquinolines and 4,5,6,7-tetrahydro-3H-imidazo[4,5-c]pyridines on a solid support has been developed. The route utilizes substituted in-tyramines, histamines and various aromatic, aliphatic and heterocyclic aldehydes. Copyright (C) 1996 Elsevier Science Ltd

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页码：4865 / 4868

页数：4

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