''Traceless'' solid-phase synthesis of furans via 1,3-dipolar cycloaddition reactions of isomunchnones

被引：65

作者：

Gowravaram, MR ^{[1
]}

Gallop, MA ^{[1
]}

机构：

[1] AFFYMAX RES INST,PALO ALTO,CA 94304

来源：

TETRAHEDRON LETTERS | 1997年 / 38卷 / 40期

关键词：

D O I：

10.1016/S0040-4039(97)01667-5

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The generation and cycloaddition reactions of polymer-supported mesoionic isomunchnones derived from alpha-diazocarbonyl intermediates is described in this report. This chemistry provides a method for preparing combinatorial libraries of functionalized furans and features cycloreversion as a new synthetic strategy for ''traceless'' synthesis of small organic molecules. (C) 1997 Elsevier Science Ltd.

引用

页码：6973 / 6976

页数：4

共 33 条

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