An efficient copper-catalyzed coupling reaction of pyridin-2-ones with aryl and heterocyclic halides based on Buchwald's protocol

被引：48

作者：

Li, CS ^{[1
]}

Dixon, DD ^{[1
]}

机构：

[1] Merck Frosst Canada Inc, Merck Frosst Ctr Therapeut Res, Pointe Claire, PQ H9R 4P8, Canada

来源：

TETRAHEDRON LETTERS | 2004年 / 45卷 / 22期

关键词：

pyridin-2-ones; aryl halides; copper-catalyzed coupling reaction;

D O I：

10.1016/j.tetlet.2004.04.019

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

An efficient copper-catalyzed coupling reaction based on the Buchwald's protocol has been established for pyridin-2-ones with aryl iodides, aryl bromides, and heterocyclic bromides. (C) 2004 Elsevier Ltd. All rights reserved.

引用

页码：4257 / 4260

页数：4

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