Isosteric replacement of acidic with neutral residues in extracellular loop-2 of the κ-opioid receptor does not affect dynorphin A(1-13) affinity and function

被引：16

作者：

Ferguson, DM

Kramer, S

Metzger, TG

Law, PY

Portoghese, PS ^{[1
]}

机构：

[1] Univ Minnesota, Coll Pharm, Dept Med Chem, Minneapolis, MN 55455 USA

[2] Univ Minnesota, Sch Med, Dept Pharmacol, Minneapolis, MN 55455 USA

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 2000年 / 43卷 / 07期

关键词：

D O I：

10.1021/jm990583r

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1251 / 1252

页数：2

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