1-(Phenylsulfonyl)indol-2-yl triflate: A versatile reagent for the synthesis of 2-substituted indoles.

被引：18

作者：

Joseph, B ^{[1
]}

Malapel, B ^{[1
]}

Merour, JY ^{[1
]}

机构：

[1] UNIV ORLEANS,INST CHIM ORGAN & ANALYT,F-45067 ORLEANS 02,FRANCE

来源：

SYNTHETIC COMMUNICATIONS | 1996年 / 26卷 / 17期

关键词：

D O I：

10.1080/00397919608004639

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The palladium-catalysed reaction of 1-(phenyl sulfonyl)indol-2-yl triflate 1 with a variety of aryl and heteroaryl boronic acids 2 or vinyl tributylstannane 3 provides a general and an efficient method for the synthesis of 2-substituted indoles 4.

引用

页码：3289 / 3295

页数：7

共 19 条

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[J]. SYNTHETIC COMMUNICATIONS, 1992, 22 (15) : 2129 - 2141
[9] PALLADIUM-CATALYZED REACTIONS IN THE SYNTHESIS OF 3-SUBSTITUTED AND 4-SUBSTITUTED INDOLES .4.
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